SCHEMBL4688019

SCHEMBL4688019

COc1c(OCc2ccccc2)ccnc1C=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.43
ADRA1D P25100 2/20 0.43
ADRA1A P35348 2/20 0.43
ADRA1B P35368 2/20 0.43
PDCD1 Q15116 1/20 0.43
CD274 Q9NZQ7 1/20 0.43
MAPT P10636 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
ERN1 O75460 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CCNB2 O95067 1/20 0.42
CDK1 P06493 1/20 0.42
CDK4 P11802 1/20 0.42
CCNB1 P14635 1/20 0.42
CCND1 P24385 1/20 0.42
CCNB3 Q8WWL7 1/20 0.42
MAPK1 P28482 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4903979 0.90 MAPT (0.46) HTR1AADRA1DADRA1AADRA1BMAPT
SCHEMBL9237762 0.89 BCHE (0.49) HTR1AADRA1DADRA1AADRA1BL3MBTL1
SCHEMBL4157654 0.88 ABCB1 (0.49) HTR1AADRA1DADRA1AADRA1BNPC1
SCHEMBL15088139 0.81 HTR1A (0.38) HTR1AADRA1DADRA1AADRA1BMAPT
SCHEMBL30963127 0.80 ALDH1A1 (0.37) PDCD1CD274MAPTL3MBTL1ERN1
SCHEMBL4111524 0.80 ALDH1A1 (0.37) PDCD1CD274MAPTL3MBTL1ERN1
SCHEMBL4688192 0.79 L3MBTL1 (0.50) HTR1AADRA1DADRA1AADRA1BMAPT
SCHEMBL1178876 0.77 LTA4H (0.58) HTR1AMAPTL3MBTL1NPC1RAB9A
SCHEMBL4681700 0.77 RXRA (0.50) HTR1AADRA1DADRA1AADRA1BNPC1
SCHEMBL4684239 0.77 MGAM (0.44) HTR1AADRA1DADRA1AADRA1BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973906-A1 HYDROXYDIHYDROPYRIDOPY RAZINE-1,8-DIONES AND METHODS FOR INHIBITING HIV INTEGRASE Virochem Pharma Inc. (CA) 2008-10-01 EP disclosed
WO-2006066414-A1 HYDROXYDIHYDROPYRIDOPY RAZINE-1,8-DIONES AND METHODS FOR INHIBITING HIV INTEGRASE VIROCHEM PHARMA INC. (CA) 2006-06-29 WO disclosed