SCHEMBL4690843

SCHEMBL4690843

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4ccc(C(F)(F)F)cc4)CC3C2)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MGLL Q99685 1/20 0.39
SLC6A4 P31645 2/20 0.39
HRH3 Q9Y5N1 1/20 0.39
HPGD P15428 2/20 0.38
MEN1 O00255 1/20 0.38
TSHR P16473 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP3A4 P08684 1/20 0.38
DPP4 P27487 1/20 0.38
NPY2R P49146 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
EPHX2 P34913 1/20 0.37
CNR1 P21554 2/20 0.37
PRLHR P49683 2/20 0.37
PREP P48147 1/20 0.36
SLC9A1 P19634 1/20 0.35
TACR1 P25103 1/20 0.35
HSD11B1 P28845 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694154 0.90 LMNA (0.43) MGLLHPGDKMT2ANPY2RHSD11B1
SCHEMBL4695755 0.90 TACR1 (0.36) GAATSHRCNR1TACR1
SCHEMBL4695972 0.89 CHRNB2 (0.40) GAAHPGDKMT2ACYP3A4
SCHEMBL4691879 0.88 HSD11B1 (0.36) MGLLHPGDDPP4TACR1HSD11B1
SCHEMBL4691228 0.88 HSD11B1 (0.38) MGLLHPGDDPP4SLC9A1TACR1
SCHEMBL4692070 0.86 HPGD (0.36) HPGD
SCHEMBL4689519 0.86 ALDH1A1 (0.47) GAAMGLLHPGDMEN1KMT2A
SCHEMBL4690534 0.85 LMNA (0.39) HPGDKMT2ACYP3A4SLC9A1
SCHEMBL4693590 0.85 KDM1A (0.48)
SCHEMBL4693016 0.84 MGLL (0.39) MGLLNPY2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed