SCHEMBL4690534

SCHEMBL4690534

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4ccc(S(C)(=O)=O)cc4)CC3C2)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.37
CNR2 P34972 7/20 0.36
HPGD P15428 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ITGB2 P05107 1/20 0.35
ICAM1 P05362 1/20 0.35
ITGAL P20701 1/20 0.35
CYP3A4 P08684 1/20 0.35
SLC9A1 P19634 1/20 0.35
PTGS2 P35354 1/20 0.35
TNF P01375 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695961 0.89 HCRTR1 (0.36) KMT2ATNF
SCHEMBL4695972 0.87 CHRNB2 (0.40) KMT2AHPGDCYP3A4TNF
SCHEMBL4692070 0.86 HPGD (0.36) LMNACNR2HPGDTNF
SCHEMBL4689519 0.86 ALDH1A1 (0.47) LMNAKMT2AHPGDTNF
SCHEMBL4690843 0.85 GAA (0.41) KMT2AHPGDCYP3A4SLC9A1
SCHEMBL4693590 0.85 KDM1A (0.48)
SCHEMBL4696301 0.84 LMNA (0.42) LMNASLC9A1TNF
SCHEMBL4694328 0.83 TNF (0.35) KMT2ACNR2HPGDTNF
SCHEMBL4691641 0.83 CHRNB2 (0.43) KMT2AHPGDL3MBTL1TNF
SCHEMBL4690544 0.82 L3MBTL1 (0.35) CNR2HPGDL3MBTL1TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed