SCHEMBL4692415

SCHEMBL4692415

NC(=O)c1ccccc1[CH]CCN1CC2CN(C(=O)c3cc4ccccc4o3)C[C@@H]2C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.49
HRH4 Q9H3N8 1/20 0.46
MAPT P10636 2/20 0.46
POLB P06746 1/20 0.46
ALDH1A1 P00352 5/20 0.45
L3MBTL1 Q9Y468 3/20 0.45
HPGD P15428 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
NPC1 O15118 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
GRIN2B Q13224 1/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
DRD2 P14416 2/20 0.41
DRD3 P35462 2/20 0.41
GLA P06280 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4693659 0.83 CHRNB2 (0.47) RAB9AMAPTPOLBALDH1A1SMN1; SMN2
SCHEMBL4694455 0.81 CHRNB2 (0.44) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL4691846 0.80 DPP4 (0.46) HRH4L3MBTL1CA12CA1CA2
SCHEMBL4695594 0.80 HCRTR1 (0.36) DRD2DRD3
SCHEMBL4691339 0.80 AKR1C3 (0.49) HRH4POLBSMN1; SMN2CA12CA1
SCHEMBL4689903 0.80 P2RX7 (0.41) RAB9APOLBALDH1A1HPGDMEN1
SCHEMBL4690222 0.78 CHRNA4 (0.46) MAPTPOLBALDH1A1MEN1KMT2A
SCHEMBL4691301 0.78 HCRTR1 (0.44)
SCHEMBL4691802 0.78 CCR5 (0.48) RAB9AALDH1A1HPGDSMN1; SMN2NPC1
SCHEMBL4691673 0.78 HCRTR1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed