SCHEMBL4694264

SCHEMBL4694264

NC(=O)c1ccccc1[CH]CCN1CC2CN(C(=O)c3sccc3Cl)C[C@@H]2C1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
HCRTR1 O43613 11/20 0.36
HCRTR2 O43614 11/20 0.36
CCR5 P51681 2/20 0.34
HRH2 P25021 1/20 0.33
HRH1 P35367 1/20 0.33
ACHE P22303 1/20 0.31
MAPK8 P45983 1/20 0.31
SLC6A1 P30531 2/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4689903 0.86 P2RX7 (0.41) ALDH1A1CCR5SLC6A1
SCHEMBL4691802 0.84 CCR5 (0.48) ALDH1A1HCRTR1HCRTR2CCR5ACHE
SCHEMBL4694455 0.81 CHRNB2 (0.44) ALDH1A1CCR5
SCHEMBL4694336 0.80 HCRTR1 (0.36) ALDH1A1HCRTR1HCRTR2CCR5
SCHEMBL3284141 0.80 CCR5 (0.42) HCRTR1HCRTR2CCR5SLC6A1
SCHEMBL4695295 0.79 HSD17B10 (0.45) ALDH1A1HCRTR1HCRTR2MAPT
SCHEMBL4691301 0.78 HCRTR1 (0.44) HCRTR1HCRTR2CCR5
SCHEMBL4694309 0.78 HCRTR1 (0.39) HCRTR1HCRTR2
SCHEMBL4693059 0.77 CCR5 (0.37) ALDH1A1CCR5MAPK8SLC6A1
SCHEMBL4693659 0.77 CHRNB2 (0.47) ALDH1A1CCR5MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed