SCHEMBL4694336

SCHEMBL4694336

NC(=O)c1ccccc1[CH]CCN1CC2CN(C(=O)c3ccncc3Cl)C[C@@H]2C1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 12/20 0.36
HCRTR2 O43614 12/20 0.36
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
ALDH1A1 P00352 1/20 0.34
THRB P10828 1/20 0.34
CCR5 P51681 2/20 0.34
KCNK3 O14649 2/20 0.33
KCNK9 Q9NPC2 2/20 0.33
NAMPT P43490 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4689903 0.89 P2RX7 (0.41) ALDH1A1THRBCCR5
SCHEMBL4691802 0.83 CCR5 (0.48) HCRTR1HCRTR2ALDH1A1CCR5
SCHEMBL4695117 0.82 HDAC3 (0.41) HCRTR1HCRTR2NAMPT
SCHEMBL4694289 0.81 HCRTR1 (0.51) HCRTR1HCRTR2
SCHEMBL4694309 0.81 HCRTR1 (0.39) HCRTR1HCRTR2
SCHEMBL4694455 0.81 CHRNB2 (0.44) ALDH1A1CCR5
SCHEMBL4694264 0.80 ALDH1A1 (0.36) HCRTR1HCRTR2ALDH1A1CCR5
SCHEMBL3284141 0.79 CCR5 (0.42) HCRTR1HCRTR2CCR5KCNK3KCNK9
SCHEMBL4693059 0.79 CCR5 (0.37) ALDH1A1CCR5KCNK3KCNK9
SCHEMBL4694466 0.78 RIPK2 (0.50) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed