SCHEMBL4699525

SCHEMBL4699525

Cc1nsc(N(CC#N)[C@@H](CC(C)C)C(N)=O)c1-c1ccc(-c2ccncc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSL P07711 4/20 0.38
CTSS P25774 4/20 0.38
CTSB P07858 4/20 0.38
CTSK P43235 3/20 0.38
AAK1 Q2M2I8 14/20 0.37
CHEK1 O14757 1/20 0.34
GSK3B P49841 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34
BMP2K Q9NSY1 1/20 0.34
CYP3A4 P08684 1/20 0.32
NEK2 P51955 1/20 0.32
PLK1 P53350 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4701632 0.91 FNTA (0.34)
SCHEMBL4701440 0.91 CTSL (0.40) CTSLCTSSCTSBCTSKMKNK1
SCHEMBL4703027 0.89 CTSK (0.31) CTSLCTSSCTSBCTSK
SCHEMBL4701995 0.87 CTSK (0.37) CTSLCTSSCTSBCTSK
SCHEMBL4705219 0.86 F11 (0.32)
SCHEMBL4699905 0.84 CTSS (0.41) CTSLCTSSCTSBCTSKAAK1
SCHEMBL4703327 0.83 CTSL (0.46) CTSLCTSSCTSBCTSK
SCHEMBL4701807 0.83 TGFBR1 (0.36) CTSLCTSSCTSBCTSK
SCHEMBL4703250 0.83 CTSL (0.46) CTSLCTSSCTSBCTSK
SCHEMBL4701334 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed