SCHEMBL4701440

SCHEMBL4701440

Cc1nsc(N(CC#N)[C@@H](CC(C)C)C(N)=O)c1-c1ccc(-c2cccnc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSL P07711 4/20 0.40
CTSK P43235 4/20 0.40
CTSS P25774 3/20 0.40
MKNK1 Q9BUB5 6/20 0.36
MKNK2 Q9HBH9 6/20 0.36
GPR88 Q9GZN0 1/20 0.35
CTSB P07858 1/20 0.35
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
DYRK1A Q13627 1/20 0.34
SYK P43405 1/20 0.33
CYP11B2 P19099 1/20 0.33
LRRK2 Q5S007 1/20 0.33
RXFP1 Q9HBX9 1/20 0.32
NTSR1 P30989 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4699525 0.91 CTSL (0.38) CTSLCTSKCTSSMKNK1CTSB
SCHEMBL4701632 0.86 FNTA (0.34)
SCHEMBL4703027 0.84 CTSK (0.31) CTSLCTSKCTSSCTSB
SCHEMBL4705219 0.83 F11 (0.32)
SCHEMBL4701995 0.83 CTSK (0.37) CTSLCTSKCTSSCTSBLMNA
SCHEMBL4699905 0.79 CTSS (0.41) CTSLCTSKCTSSCTSBSYK
SCHEMBL4698340 0.79
SCHEMBL4701807 0.78 TGFBR1 (0.36) CTSLCTSKCTSSCTSB
SCHEMBL4703327 0.78 CTSL (0.46) CTSLCTSKCTSSCTSB
SCHEMBL4703250 0.78 CTSL (0.46) CTSLCTSKCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed