SCHEMBL4699642

SCHEMBL4699642

CC(C)C[C@@H](C(N)=O)N(CC#N)c1cscc1-c1ccc(N2CCNCC2)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSL P07711 10/20 0.44
CTSS P25774 10/20 0.44
CTSB P07858 9/20 0.44
CTSK P43235 8/20 0.44
ACVR1 Q04771 1/20 0.34
MAP2 P11137 2/20 0.33
FFAR4 Q5NUL3 1/20 0.33
JAK2 O60674 1/20 0.33
BRD4 O60885 1/20 0.33
MAPT P10636 1/20 0.32
SLC6A9 P48067 1/20 0.32
KCNH2 Q12809 1/20 0.32
MAPKAPK2 P49137 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705295 0.84 CTSL (0.45) CTSLCTSSCTSBCTSK
SCHEMBL4701371 0.81 CTSL (0.33) CTSLCTSSCTSBCTSK
SCHEMBL4700109 0.78 CTSL (0.38) CTSLCTSSCTSBCTSK
SCHEMBL4699567 0.77 CTSK (0.44) CTSLCTSSCTSBCTSK
SCHEMBL4703612 0.76 CTSS (0.34) CTSLCTSSCTSBCTSK
SCHEMBL4701830 0.76 CTSK (0.37) CTSLCTSSCTSBCTSK
SCHEMBL6801548 0.75 CTSS (0.35) CTSLCTSSCTSBCTSK
SCHEMBL4703746 0.75 OPRM1 (0.37) CTSLCTSSCTSBCTSK
SCHEMBL4699645 0.75 CTSL (0.77) CTSLCTSSCTSBCTSK
SCHEMBL4756631 0.74 RET (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed