SCHEMBL4739255

SCHEMBL4739255

COC1CN(C(=O)c2cc3c(nc(C)n3C)c3c2CCC2(Cc4ccccc4C2)O3)C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
RIPK1 Q13546 1/20 0.34
GABRA5 P31644 1/20 0.33
HCRTR1 O43613 3/20 0.33
HCRTR2 O43614 3/20 0.33
SPR P35270 1/20 0.33
RORC P51449 3/20 0.32
PDK2 Q15119 1/20 0.32
PARP1 P09874 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
TTK P33981 1/20 0.30
CCR1 P32246 1/20 0.30
CNR1 P21554 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4734384 0.87 KMT2A (0.36) SPRMEN1KMT2ACNR1
SCHEMBL4738609 0.83 DHODH (0.36) MEN1KMT2A
SCHEMBL4739107 0.81 ALDH1A1 (0.31)
SCHEMBL4737019 0.81 BACE1 (0.31) HCRTR1HCRTR2SPRRORC
SCHEMBL4737070 0.81 ALDH1A1 (0.36) GABRA5ADORA3MEN1KMT2A
SCHEMBL4739802 0.81 NPC1 (0.32)
SCHEMBL4782354 0.81 KDM4E (0.32) KMT2A
SCHEMBL4737882 0.80 RAB9A (0.35) RIPK1KMT2ACCR1CNR1CNR2
SCHEMBL4734073 0.79 CHIA (0.33)
SCHEMBL4739132 0.78 KDM4E (0.40) RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071765-A1 PHARMACEUTICALLY ACTIVE SPIRO-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-06-19 WO claimed