SCHEMBL4739877

SCHEMBL4739877

O=C(O)CC1CCCN(S(=O)(=O)c2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
CYP19A1 P11511 2/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C19 P33261 1/20 0.50
RAB9A P51151 3/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
GAA P10253 2/20 0.48
HTT P42858 1/20 0.48
NPC1 O15118 1/20 0.47
ATM Q13315 1/20 0.47
AKR1C3 P42330 4/20 0.47
AKR1C1 Q04828 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
KDM4E B2RXH2 1/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4741097 0.85 ALDH1A1 (0.51) TSHRCYP19A1CYP3A4CYP2C19RAB9A
SCHEMBL4740459 0.85 ALDH1A1 (0.51) TSHRCYP19A1CYP3A4CYP2C19RAB9A
SCHEMBL4741043 0.85 KMT2A (0.58) CYP19A1CYP3A4CYP2C19GAAHTT
SCHEMBL4740625 0.82 LMNA (0.57) TSHRCYP3A4CYP2C19L3MBTL1HTT
SCHEMBL643115 0.78 HTR7 (0.60) TSHRCYP3A4CYP2C19L3MBTL1GAA
SCHEMBL4741083 0.78 TSHR (0.58) TSHRAKR1C3AKR1C1KMT2AKDM4E
SCHEMBL7697945 0.77 CHRM5 (0.51) CYP2C19RAB9AGAAHTT
SCHEMBL4739879 0.77 RAB9A (0.58) RAB9AGAAHTTMEN1KMT2A
SCHEMBL5500815 0.77 AKR1C3 (0.41) TSHRCYP19A1CYP3A4CYP2C19RAB9A
SCHEMBL4740463 0.77 TSHR (0.56) TSHRAKR1C3AKR1C1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087654-A2 PIPERIDINES AS INHIBITORS OF 11β-HYDROXYSTEROID DEHYDROGENASE TYPE 1 CADILA HEALTHCARE LIMITED (IN) 2008-07-24 WO disclosed