SCHEMBL474101

SCHEMBL474101

COC(=O)c1ccc(Cl)nn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.47
JUN P05412 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
NOTUM Q6P988 2/20 0.42
KMT2A Q03164 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MEN1 O00255 2/20 0.42
KDM4E B2RXH2 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
LMNA P02545 1/20 0.40
NNMT P40261 1/20 0.40
ALDH1A1 P00352 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29552833 1.00 MAPK1 (0.47) MAPK1JUNNFKB1NFKB2RELA
SCHEMBL1456298 0.87 MAPK1 (0.57) MAPK1NOTUMKMT2AMEN1KDM4E
SCHEMBL29442775 0.87 MAPK1 (0.57) MAPK1NOTUMKMT2AMEN1KDM4E
SCHEMBL30670211 0.79 LMNA (0.55) JUNNFKB1NFKB2RELAKMT2A
SCHEMBL26657700 0.79 ALDH1A1 (0.44) JUNNFKB1NFKB2RELAKMT2A
SCHEMBL2473041 0.79 CYP1A2 (0.53) NOTUMKMT2AMEN1KDM4EL3MBTL1
SCHEMBL20046201 0.79 LMNA (0.55) JUNNFKB1NFKB2RELAKMT2A
SCHEMBL18979849 0.79 KDM4E (0.56) MAPK1KDM4EL3MBTL1NNMTALDH1A1
SCHEMBL31058092 0.79 MAPK1 (0.50) MAPK1NOTUMKMT2AMEN1KDM4E
SCHEMBL14966683 0.79 MAPK1 (0.50) MAPK1NOTUMKMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 563 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118598859-A Nitrogenous heterocyclic indole xanthine oxidase inhibitor and preparation method and application thereof 武汉工程大学 2024-09-06 CN claimed
CN-118515650-A STING agonist A02 and synthetic method and application thereof 河南牧业经济学院 2024-08-20 CN claimed
CN-118440058-A N-phenylpyridazine-3-carboxamide compound as well as preparation method and application thereof 武汉大学深圳研究院 2024-08-06 CN claimed
US-12637468-B2 Substituted [1,2,4]triazolo[4,3-b]pyridazines as GABAA receptor modulators Shanghai Simr Biotechnology Co., Ltd. (CN) 2026-05-26 US disclosed
US-20260132111-A1 Host-Targeted Pan-Respiratory Antiviral Small Molecule Therapeutics PROSETTA BIOSCIENCES INC (US) 2026-05-14 US disclosed
EP-4727922-A1 DUAL RAF AND TUBULIN INHIBITORS AND METHODS OF USE THEREOF Deciphera Pharmaceuticals, LLC (US) 2026-04-22 EP disclosed
US-20260053796-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR ARVINAS OPERATIONS INC (US) 2026-02-26 US disclosed
US-20260035384-A1 COMPOUND CONTAINING CYCLOHEXYL CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD (CN) 2026-02-05 US disclosed
US-20260035361-A1 COMPOUNDS FOR MODULATING HUR (ELAVL1) SHANGHAI DEGRON BIOMEDICAL TECH CO LTD (CN) 2026-02-05 US disclosed
EP-3755331-B1 AGONISTS OF STIMULATOR OF INTERFERON GENES (STING) FOR USE IN THE TREATMENT OF CANCER SCRIPPS RESEARCH INST (US) 2026-01-28 EP disclosed
US-20260014147-A1 STAT6 DEGRADERS GILEAD SCIENCES INC (US) 2026-01-15 US disclosed
WO-2005028452-A1 SUBSTITUTED TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-03-31 WO disclosed
US-20050065143-A1 Pyridazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2005-03-24 US disclosed
WO-2005011655-A2 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2005-02-10 WO disclosed
US-20040152699-A1 Compounds ASTRAZENECA AND NPS PHARMACEUTICALS, INC. 2004-08-05 US disclosed
WO-2004026305-A9 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONIST LILLY CO ELI (US) 2004-05-13 WO disclosed
WO-2004026305-A1 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONIST ELI LILLY AND COMPANY (US) 2004-04-01 WO disclosed
WO-2004014881-A2 '1,2,4'OXADIAZOLES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR-5 ASTRA ZENECA AB (SE) 2004-02-19 WO disclosed
US-5340808-A Fused pyridazinoquinazolone derivatives as neurotrophic agents WARNER LAMBERT COMPANY (US) 1994-08-23 US disclosed
WO-1994011373-A1 PYRIDAZINOQUINAZOLONE DERIVATIVES AS NEUROTROPHIC AGENTS WARNER-LAMBERT COMPANY (US) 1994-05-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040152699-A1 Compounds SDHA, CYP11B2, CYP11B1 MAPK1 2417/4885JUN 3270/4885NFKB1 656/4885
US-20050065143-A1 Pyridazine derivatives and their use as therapeutic agents PRDX5, SNRPD3, SNRPD2 MAPK1 3803/4885JUN 4855/4885NFKB1 2224/4885
US-20260132111-A1 Host-Targeted Pan-Respiratory Antiviral Small Molecule Therapeutics NCOR1, HAVCR2, NR3C1 MAPK1 3571/4885JUN 2510/4885NFKB1 3290/4885
US-20260053796-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR AR, NR5A1, KLK3 MAPK1 2144/4885JUN 4119/4885NFKB1 2961/4885
US-12637468-B2 Substituted [1,2,4]triazolo[4,3-b]pyridazines as GABAA receptor modulators GABRA6, GABRA1, GABRB1 MAPK1 2422/4885JUN 2262/4885NFKB1 3370/4885
US-20260035384-A1 COMPOUND CONTAINING CYCLOHEXYL CYP11B1, CYP4A11, CYP11B2 MAPK1 3002/4885JUN 2750/4885NFKB1 1211/4885
US-20260014147-A1 STAT6 DEGRADERS STAT6, NCOR1, CBR1 MAPK1 2558/4885JUN 1586/4885NFKB1 1548/4885
US-20260035361-A1 COMPOUNDS FOR MODULATING HUR (ELAVL1) ELAVL1, ELAVL3, HNRNPL MAPK1 3753/4885JUN 997/4885NFKB1 1858/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.