SCHEMBL4754290

SCHEMBL4754290

CC1(C)Cc2cc(N)cc(OCCN3CCN(c4cccc(C(F)(F)F)c4)CC3)c2O1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.50
MAPT P10636 2/20 0.50
ALDH1A1 P00352 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
MAPK1 P28482 1/20 0.50
CYP2C19 P33261 1/20 0.50
THPO P40225 1/20 0.50
MTOR P42345 1/20 0.50
BLM P54132 1/20 0.50
PMP22 Q01453 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
ABCB1 P08183 3/20 0.49
HTR4 Q13639 1/20 0.48
HTR7 P34969 1/20 0.48
DRD2 P14416 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4751067 0.86 HTR7 (0.47) HTR1AALDH1A1SMN1; SMN2ABCB1HTR4
SCHEMBL4752802 0.84 ALDH1A1 (0.41) HTR1AALDH1A1SMN1; SMN2ABCB1HTR4
SCHEMBL4908879 0.83 HTR7 (0.50) HTR1AABCB1HTR7DRD2HTR2A
SCHEMBL4788339 0.82 KCNH2 (0.50) ABCB1HTR4SIGMAR1HTR2A
SCHEMBL4754299 0.80 ADRA1A (0.41) HTR1AALDH1A1SMN1; SMN2ABCB1HTR7
Hydrochloric Acid SCHEMBL4788931 0.76 GAA (0.53) MAPTALDH1A1TSHRMAPK1SMN1; SMN2
SCHEMBL4863289 0.71 ALDH1A1 (0.41) HTR1AMAPTALDH1A1CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL4789017 0.70 KCNH2 (0.49) ABCB1SIGMAR1HTR2A
SCHEMBL314513 0.70 ALDH1A1 (0.64) ALDH1A1CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL11810344 0.70 HTR2A (0.62) HTR1AMAPTALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008146063-A1 NEW BENZOFURAN DERIVATIVES AS SELECTIVE 5HT6 RECEPTOR INHIBITORS AND PROCESS FOR THEIR PREPARATION EGIS GYÓGYSZERGYÁR Nyilvánosan Müködö Részvénytársagág (HU) 2008-12-04 WO disclosed