SCHEMBL4752802

SCHEMBL4752802

COc1ccc(C(F)(F)F)cc1N1CCN(CCOc2cc(N)cc3c2OC(C)(C)C3)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
HTR1A P08908 5/20 0.40
HTR1B P28222 2/20 0.40
ADRA1A P35348 2/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1B P35368 1/20 0.40
HTR4 Q13639 1/20 0.38
HTR2C P28335 4/20 0.38
HTR2A P28223 4/20 0.38
HTR6 P50406 3/20 0.38
HTR1D P28221 1/20 0.38
ABCB1 P08183 1/20 0.37
MCHR1 Q99705 1/20 0.36
DRD2 P14416 1/20 0.36
HTR7 P34969 1/20 0.36
CACNA1G O43497 1/20 0.36
KCNH2 Q12809 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4754299 0.96 ADRA1A (0.41) ALDH1A1SMN1; SMN2FFAR4HTR1AHTR1B
SCHEMBL4863289 0.87 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2FFAR4HTR1AHTR1B
SCHEMBL4754290 0.84 HTR1A (0.50) ALDH1A1SMN1; SMN2HTR1AHTR4HTR2A
SCHEMBL4751067 0.71 HTR7 (0.47) ALDH1A1SMN1; SMN2HTR1AHTR4HTR2A
SCHEMBL12969072 0.71 HTR6 (0.58) ALDH1A1FFAR4HTR1AHTR1BADRA1A
SCHEMBL4788339 0.70 KCNH2 (0.50) HTR4HTR2AABCB1KCNH2
SCHEMBL28496894 0.69 KMT2A (0.39) ALDH1A1HTR2AKDM4E
SCHEMBL28978441 0.69 DHFR (0.40) ALDH1A1HTR1AHTR2AKDM4E
SCHEMBL4908879 0.68 HTR7 (0.50) HTR1AHTR2CHTR2AHTR6ABCB1
SCHEMBL4753309 0.68 NPC1 (0.37) ALDH1A1FFAR4HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008146063-A1 NEW BENZOFURAN DERIVATIVES AS SELECTIVE 5HT6 RECEPTOR INHIBITORS AND PROCESS FOR THEIR PREPARATION EGIS GYÓGYSZERGYÁR Nyilvánosan Müködö Részvénytársagág (HU) 2008-12-04 WO disclosed