SCHEMBL475565

SCHEMBL475565

COC(=O)c1ccnc(C(=O)O)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.68
KDM6B O15054 2/20 0.68
KDM5C P41229 2/20 0.68
KDM4C Q9H3R0 2/20 0.68
KDM2A Q9Y2K7 2/20 0.68
KDM3A Q9Y4C1 2/20 0.68
ALDH1A1 P00352 5/20 0.67
MAPT P10636 3/20 0.67
KDM5B Q9UGL1 2/20 0.67
ALKBH5 Q6P6C2 2/20 0.67
FTO Q9C0B1 2/20 0.67
TET3 O43151 1/20 0.67
KDM4A O75164 1/20 0.67
BBOX1 O75936 1/20 0.67
KDM5A P29375 1/20 0.67
ASPH Q12797 1/20 0.67
KDM4D Q6B0I6 1/20 0.67
TET2 Q6N021 1/20 0.67
KDM7A Q6ZMT4 1/20 0.67
KDM8 Q8N371 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30779113 1.00 KDM4E (0.68) KDM4EKDM6BKDM5CKDM4CKDM2A
SCHEMBL70350 0.89 KDM4E (0.62) KDM4EKDM6BKDM5CKDM4CKDM2A
SCHEMBL30065796 0.89 KDM4E (0.62) KDM4EKDM6BKDM5CKDM4CKDM2A
SCHEMBL30745026 0.86 KDM4E (0.68) KDM4EKDM6BKDM5CKDM4CKDM2A
SCHEMBL2716237 0.86 KDM4E (0.68) KDM4EKDM6BKDM5CKDM4CKDM2A
SCHEMBL30378954 0.86 KDM4E (0.58) KDM4EKDM6BKDM5CKDM4CKDM2A
SCHEMBL1759313 0.86 KDM4E (0.58) KDM4EKDM6BKDM5CKDM4CKDM2A
SCHEMBL13950719 0.84 KDM4E (0.57) KDM4EKDM6BKDM5CKDM4CKDM2A
SCHEMBL1759324 0.84 KDM4E (0.57) KDM4EKDM6BKDM5CKDM4CKDM2A
SCHEMBL19616007 0.83 KDM4E (0.60) KDM4EKDM6BKDM5CKDM4CKDM2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 78 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103788079-A Preparation method for isonicotinic acid WUXI VISION PRO LTD 2014-05-14 CN claimed
CN-112707873-B Substituted oxazole derivative and application thereof in medicines 广东东阳光药业股份有限公司 2023-12-08 CN disclosed
US-11807886-B2 Process for the preparation of copolymers derived from 2,4- or 2,5-pyridinedicarboxylic acid BIOME BIOPLASTICS LIMITED (GB) 2023-11-07 US disclosed
US-20230212190-A1 PROBES FOR IMAGING HUNTINGTIN PROTEIN CHDI FOUNDATION, INC. 2023-07-06 US disclosed
US-20230212190-A1 PROBES FOR IMAGING HUNTINGTIN PROTEIN CHDI FOUNDATION, INC. 2023-07-06 US disclosed
EP-3307901-B1 PROCESS FOR THE PREPARATION OF 2,4- OR 2,5-PYRIDINEDICARBOXYLIC ACID BIOME BIOPLASTICS LTD (GB) 2022-04-27 EP disclosed
US-11059836-B2 Probes for imaging huntingtin protein CHDI FOUNDATION, INC. (US) 2021-07-13 US disclosed
US-20210206963-A1 COPOLYMER BLENDS BIOME BIOPLASTICS LIMITED (GB) 2021-07-08 US disclosed
US-10612057-B2 Process for the preparation of 2,4- or 2,5-pyridinedicarboxylic acid and copolymers derived therefrom BIOME BIOPLASTICS LIMITED (GB) 2020-04-07 US disclosed
WO-2020035593-A1 COPOLYMER BLENDS BIOME BIOPLASTICS LIMITED (GB) 2020-02-20 WO disclosed
US-20070082900-A1 Methods for inhibiting protein kinases SCHERING CORPORATION 2007-04-12 US disclosed
US-20070072881-A1 Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors SCHERING CORPORATION 2007-03-29 US disclosed
EP-0585328-B1 SUBSTITUTED 3-AMINOQUINUCLIDINES PFIZER (US) 2002-01-09 EP disclosed
US-5852038-A Substituted 3-aminoquinuclidines PFIZER INC (US) 1998-12-22 US disclosed
US-5716965-A Substituted 3-aminoquinuclidines PFIZER INC. (US) 1998-02-10 US disclosed
EP-0533132-B1 Process for the oxidation of hydroxymethylpyridine derivatives to pyridine carboxylic acid derivatives HOECHST AG (DE) 1994-11-02 EP disclosed
EP-0585328-A1 SUBSTITUTED 3-AMINOQUINUCLIDINES PFIZER INC. (US) 1994-03-09 EP disclosed
US-5259933-A Process for oxidizing hydroxymethylpyridine derivatives to pyridinecarboxylic acid derivatives at nickel oxide hydroxide anodes HOECHST AKTIENGESELLSCHAFT (DE) 1993-11-09 US disclosed
EP-0533132-A1 Process for the oxidation of hydroxymethylpyridine derivatives to pyridine carboxylic acid derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1993-03-24 EP disclosed
WO-1992020676-A1 SUBSTITUTED 3-AMINOQUINUCLIDINES PFIZER INC. (US) 1992-11-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230212190-A1 PROBES FOR IMAGING HUNTINGTIN PROTEIN HTT, HYPK, HSPBP1 KDM4E 4585/4885KDM6B 4697/4885KDM5C 4770/4885
US-20070082900-A1 Methods for inhibiting protein kinases PIM1, AURKC, PIM3 KDM4E 1092/4885KDM6B 1334/4885KDM5C 762/4885
US-11807886-B2 Process for the preparation of copolymers derived from 2,4- or 2,5-pyridinedicarboxylic acid HPD, PGD, PCCA KDM4E 378/4885KDM6B 647/4885KDM5C 261/4885
US-11059836-B2 Probes for imaging huntingtin protein HTT, HYPK, HSPBP1 KDM4E 4585/4885KDM6B 4697/4885KDM5C 4770/4885
US-10612057-B2 Process for the preparation of 2,4- or 2,5-pyridinedicarboxylic acid and copolymers derived therefrom HPD, PCCA, MVD KDM4E 657/4885KDM6B 484/4885KDM5C 536/4885
US-20070072881-A1 Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors CDK2, CDK1, CDKN1A KDM4E 673/4885KDM6B 864/4885KDM5C 482/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.