SCHEMBL476304

SCHEMBL476304

COC(=O)C1CCC(=O)N1C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
WNT3 P56703 1/20 0.39
SFRP1 Q8N474 1/20 0.39
PTPN1 P18031 2/20 0.38
BRD4 O60885 1/20 0.37
MMP2 P08253 1/20 0.37
ANPEP P15144 1/20 0.37
MEN1 O00255 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ELANE P08246 1/20 0.35
PDE4B Q07343 1/20 0.35
ACE P12821 2/20 0.35
EPHX1 P07099 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL476303 1.00 KMT2A (0.41) KMT2ACHRM2CHRM1CHRM3WNT3
SCHEMBL540990 1.00 KMT2A (0.41) KMT2ACHRM2CHRM1CHRM3WNT3
SCHEMBL1604617 0.91 MMP2 (0.38) KMT2ACHRM2CHRM1CHRM3WNT3
SCHEMBL1604618 0.91 MMP2 (0.38) KMT2ACHRM2CHRM1CHRM3WNT3
SCHEMBL18018362 0.91 MMP2 (0.38) KMT2ACHRM2CHRM1CHRM3WNT3
SCHEMBL713924 0.91 CHRM2 (0.41) CHRM2CHRM1CHRM3WNT3SFRP1
SCHEMBL1372911 0.91 CHRM2 (0.41) CHRM2CHRM1CHRM3WNT3SFRP1
SCHEMBL12105456 0.91 CHRM2 (0.41) CHRM2CHRM1CHRM3WNT3SFRP1
SCHEMBL30289778 0.91 CHRM2 (0.41) CHRM2CHRM1CHRM3WNT3SFRP1
SCHEMBL6743320 0.88 CHRM2 (0.38) CHRM2CHRM1CHRM3WNT3SFRP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 178 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250206759-A1 FUSED RING COMPOUND, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND USE OF FUSED RING COMPOUND CHENGDU HYPERWAY PHARMACEUTICALS CO., LTD. (CN) 2025-06-26 US disclosed
US-12240869-B2 Inhibitors of cyclin-dependent kinase 7 (CDK7) SYROS PHARMACEUTICALS, INC. (US) 2025-03-04 US disclosed
EP-4509507-A1 FUSED RING COMPOUND, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND USE OF FUSED RING COMPOUND Chengdu Hyperway Pharmaceuticals Co., Ltd. (CN) 2025-02-19 EP disclosed
US-20240360165-A1 INHIBITORS OF CYCLIN DEPENDENT KINASE 7 (CDK7) MEDIC LIFE SCIENCES, INC. 2024-10-31 US disclosed
US-20240294520-A1 AMINO ACID COMPOUNDS WITH UNBRANCHED LINKERS AND METHODS OF USE PLIANT THERAPEUTICS INC (US) 2024-09-05 US disclosed
WO-2024091409-A1 TRICYCLIC DERIVATIVES AS KRAS INHIBITORS NIKANG THERAPEUTICS, INC. (US) 2024-05-02 WO disclosed
US-20240124435-A1 COMPOUNDS AND USES THEREOF JANSSEN PHARMACEUTICA NV (BE) 2024-04-18 US disclosed
CN-117777121-A Compounds and uses thereof 詹森药业有限公司 2024-03-29 CN disclosed
WO-2024054625-A2 BIFUNCTIONAL COMPOUNDS FOR DEGRADING KRAS G12D VIA UBIQUITIN PROTEASOME PATHWAY NIKANG THERAPEUTICS, INC. (US) 2024-03-14 WO disclosed
US-20240034742-A1 DOSING REGIMENS FOR CYCLIN-DEPENDENT KINASE 7 (CDK7) INHIBITORS MEDIC LIFE SCIENCES, INC. 2024-02-01 US disclosed
WO-2009023473-A2 ANTIMICROBIAL PARENTERAL FORMULATION TAIGEN BIOTECHNOLOGY CO., LTD. (TW) 2009-02-19 WO disclosed
US-20090042932-A1 ANTIMICROBIAL PARENTERAL FORMULATION TAIGEN BIOTECHNOLOGY COMPANY LTD. (TW) 2009-02-12 US disclosed
US-7456279-B2 Coupling process for preparing quinolone intermediates THE PROCTER & GAMBLE COMPANY (US) 2008-11-25 US disclosed
US-20080058528-A1 useful in the treatment of disorders mediated by DPP-IV such as, but not limited to, diabetes, type II diabetes, hyperglycemia, Syndrome X, hyperinsulinemia and obesity ABBVIE INC. 2008-03-06 US disclosed
US-7279485-B2 Substituted heterocyclic derivatives useful as antidiabetic and antiobesity agents and method BRISTOL-MYERS SQUIBB COMPANY (US) 2007-10-09 US disclosed
US-20070054842-A1 Novel macrocyclic inhibitors of hepatitis C virus replication ARRAY BIOPHARMA, INC. 2007-03-08 US disclosed
US-7041696-B2 Interleukin-1β converting enzyme inhibitors THE PROCTER & GAMBLE COMPANY (US) 2006-05-09 US disclosed
EP-1513844-A1 NOVEL INTERLEUKIN-1 BETA CONVERTING ENZYME INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2005-03-16 EP disclosed
US-20030236296-A1 Novel interleukin-1beta converting enzyme inhibitors THE PROCTER & GAMBLE COMPANY 2003-12-25 US disclosed
WO-2003106460-A1 NOVEL INTERLEUKIN-1 BETA CONVERTING ENZYME INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2003-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090042932-A1 ANTIMICROBIAL PARENTERAL FORMULATION SLC10A2, ABCB11, SLC47A1 KMT2A 4823/4885CHRM2 4147/4885CHRM1 4067/4885
US-20240034742-A1 DOSING REGIMENS FOR CYCLIN-DEPENDENT KINASE 7 (CDK7) INHIBITORS CDK7, CCNI, CDK17 KMT2A 826/4885CHRM2 4866/4885CHRM1 4728/4885
US-20240124435-A1 COMPOUNDS AND USES THEREOF NLN, ACHE, CLN6 KMT2A 2479/4885CHRM2 1129/4885CHRM1 1838/4885
US-20080058528-A1 useful in the treatment of disorders mediated by DPP-IV such as, but not limited to, diabetes, type II diabetes, hyperglycemia, Syndrome X, hyperinsulinemia and obesity DPP4, DPP7, DPP3 KMT2A 1506/4885CHRM2 2158/4885CHRM1 1676/4885
US-20070054842-A1 Novel macrocyclic inhibitors of hepatitis C virus replication EIF2AK2, HAVCR2, HCCS KMT2A 3154/4885CHRM2 4816/4885CHRM1 4813/4885
US-20240360165-A1 INHIBITORS OF CYCLIN DEPENDENT KINASE 7 (CDK7) CDK7, CDK3, CDK9 KMT2A 1277/4885CHRM2 4844/4885CHRM1 4761/4885
US-12240869-B2 Inhibitors of cyclin-dependent kinase 7 (CDK7) CDK7, CDK1, CDK17 KMT2A 2154/4885CHRM2 4793/4885CHRM1 4605/4885
US-20250206759-A1 FUSED RING COMPOUND, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND USE OF FUSED RING COMPOUND KRAS, NRAS, HRAS KMT2A 966/4885CHRM2 4374/4885CHRM1 3852/4885
US-20240294520-A1 AMINO ACID COMPOUNDS WITH UNBRANCHED LINKERS AND METHODS OF USE ITGA2B, ITGB6, ITGB1 KMT2A 1467/4885CHRM2 422/4885CHRM1 387/4885
US-20030236296-A1 Novel interleukin-1beta converting enzyme inhibitors IL1R1, IL1B, IL1RN KMT2A 3683/4885CHRM2 1812/4885CHRM1 1064/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.