SCHEMBL4789083

SCHEMBL4789083

CN1CCN(c2ccc(Br)c3c2CC(N)C(Cc2ccccc2)(Cc2ccccc2)O3)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MC4R P32245 1/20 0.35
DRD2 P14416 4/20 0.35
DRD3 P35462 4/20 0.35
DRD4 P21917 2/20 0.35
ADRA2C P18825 1/20 0.35
HTR6 P50406 5/20 0.34
HRH4 Q9H3N8 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
SIGMAR1 Q99720 2/20 0.33
TMEM97 Q5BJF2 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
MAPK1 P28482 2/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788517 0.69 L3MBTL1 (0.43) HRH4LMNAPOLBKMT2AMAPT
SCHEMBL4750457 0.65 HTR2C (0.41) HTR6SMN1; SMN2KDM4E
SCHEMBL8160398 0.65 SIGMAR1 (0.36) MC4RDRD2DRD3DRD4ADRA2C
SCHEMBL4749790 0.64 HRH1 (0.41) SMN1; SMN2LMNAKMT2AMAPTKDM4E
SCHEMBL6819394 0.64 DRD2 (0.43) DRD2DRD3KMT2ASIGMAR1TMEM97
Lithium Ion SCHEMBL4750393 0.63 SIGMAR1 (0.39) DRD2ADRA2CLMNASIGMAR1HTR1A
SCHEMBL6820056 0.62 ADRA1A (0.39) DRD2DRD3ADRA2CHTR6POLB
SCHEMBL6820067 0.62 ADRA1A (0.39) DRD2DRD3ADRA2CHTR6POLB
SCHEMBL4747515 0.62 ADRA2C (0.38) DRD2DRD3DRD4ADRA2CHTR6
SCHEMBL4787846 0.62 HRH1 (0.47) DRD2DRD3DRD4SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130321-A2 NOVEL N-TETRAHYDRONAPHTALENE OR 5-HETEROCYCLYL-CHROMANE OR 8-HETEROCYCLYL-TETRAHYDRONAPHTALENE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed