SCHEMBL4749790

SCHEMBL4749790

CN1CCC(O)CC1.CN1CCC(Oc2cccc3c2CC(N)C(Cc2ccccc2)(Cc2ccccc2)O3)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 2/20 0.41
KDM4E B2RXH2 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
NPY1R P25929 1/20 0.39
NPY2R P49146 1/20 0.39
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SCN1A P35498 2/20 0.35
SCN2A Q99250 2/20 0.35
SCN3A Q9NY46 2/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM1A O60341 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CHRM5 P08912 3/20 0.32
CHRM1 P11229 3/20 0.32
CHRM3 P20309 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4750457 0.91 HTR2C (0.41) HRH1KDM4ESMN1; SMN2NPY1RNPY2R
SCHEMBL4750969 0.86 HTR2C (0.38) HRH1HTR2CHTR2BMEN1KMT2A
SCHEMBL4787846 0.75 HRH1 (0.47) HRH1KDM4ESMN1; SMN2
SCHEMBL4788517 0.73 L3MBTL1 (0.43) KDM4EMAPTLMNAALDH1A1KDM1A
SCHEMBL4788942 0.71 GABRA1 (0.34) KDM4EMAPTKDM1AMEN1KMT2A
SCHEMBL4750047 0.69 SMN1; SMN2 (0.39) HRH1KDM4ESMN1; SMN2NPY1RNPY2R
Lithium Ion SCHEMBL4750393 0.65 SIGMAR1 (0.39) LMNANPSR1KDM1A
SCHEMBL4789083 0.64 MC4R (0.35) KDM4ESMN1; SMN2MAPTLMNAALDH1A1
SCHEMBL4747586 0.64 NOS3 (0.40) HTR2CHTR2B
SCHEMBL4786874 0.63 DRD2 (0.52) KDM4ESMN1; SMN2NPY1RNPY2RKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130319-A2 NOVEL N-TETRAHYDRONAPHTALENE OR N-CHROMANE CARBOXAMIDE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed