SCHEMBL4789529

SCHEMBL4789529

CCC(C#N)(CC1C2CCC1CN(CCc1ccc3c(c1)OCO3)C2)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.41
ADRA1D P25100 3/20 0.41
ADRA1B P35368 3/20 0.41
TSHR P16473 3/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
CHRM5 P08912 2/20 0.35
CHRM1 P11229 2/20 0.35
DRD2 P14416 2/20 0.35
CHRM3 P20309 2/20 0.35
ADRB2 P07550 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
ADRB1 P08588 1/20 0.35
ADRA2A P08913 1/20 0.35
KCNE1 P15382 1/20 0.35
ADRA2B P18089 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4789432 0.91 ADRA1D (0.42) ADRA1AADRA1DADRA1BTSHRALDH1A1
SCHEMBL4789955 0.88 TSHR (0.42) ADRA1AADRA1DADRA1BTSHRALDH1A1
SCHEMBL4789936 0.83 CHRM3 (0.33) TSHRALDH1A1KDM4EMEN1MAPK1
SCHEMBL4788488 0.82 CHRM3 (0.40) ADRA1AADRA1DADRA1BTSHRALDH1A1
SCHEMBL4789352 0.78 TSHR (0.47) TSHRKDM4EMEN1KMT2ADRD2
SCHEMBL4789381 0.78 ALDH1A1 (0.44) ADRA1AADRA1DADRA1BTSHRALDH1A1
SCHEMBL4789694 0.78 CHRM3 (0.48) ADRA1AADRA1DADRA1BTSHRALDH1A1
SCHEMBL4788351 0.77 ALDH1A1 (0.34) TSHRALDH1A1MEN1KMT2ACHRM3
SCHEMBL4758052 0.77 DRD2 (0.42) CHRM1DRD2CHRM3CHRM2DRD3
SCHEMBL4790238 0.75 ALDH1A1 (0.35) ADRA1AADRA1DTSHRALDH1A1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008117229-A1 MUSCARINIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2008-10-02 WO claimed
WO-2008117229-A1 MUSCARINIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2008-10-02 WO disclosed