SCHEMBL4841791

SCHEMBL4841791

CC(C)(C)C(O[SiH](c1ccccc1)c1ccccc1)c1cccc(C#CCCCCO)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.40
HTR2B P41595 2/20 0.40
CHRNB4 P30926 2/20 0.38
CHRNA3 P32297 2/20 0.38
EGFR P00533 2/20 0.35
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
MAPT P10636 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
KDM4E B2RXH2 1/20 0.34
BACE1 P56817 1/20 0.34
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
ATM Q13315 1/20 0.32
RCE1 Q9Y256 1/20 0.32
TSHR P16473 1/20 0.31
GABRP O00591 1/20 0.31
GABRD O14764 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5555730 0.78 ALDH1A1 (0.35) ALDH1A1KDM4ELMNA
SCHEMBL4848474 0.78 CYP4F2 (0.39)
SCHEMBL8796135 0.74 TSHR (0.34) KMT2AMEN1TSHR
SCHEMBL8149465 0.72 ADRB1 (0.41) HTR2BCYP3A4KDM4ETSHRLMNA
SCHEMBL6622199 0.70 MAOB (0.34) ALDH1A1CYP3A4MAPTKDM4EKMT2A
SCHEMBL8796366 0.70 IDO1 (0.42) ALDH1A1CYP3A4KMT2AMEN1
SCHEMBL7985829 0.69 ADRB2 (0.34) CYP1A2TSHR
SCHEMBL8795978 0.69 TRPA1 (0.32)
SCHEMBL8794946 0.69 ENPP2 (0.35) KDM4E
SCHEMBL4841777 0.69 HTR2C (0.43) HTR2CHTR2BCHRNB4CHRNA3EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE40558-E1 Therapeutic uses of di-aryl acid derivatives SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2008-10-28 US disclosed
US-6635655-B1 Agonists or antagonists of peroxisome proliferator-activated receptors AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-10-21 US disclosed
EP-1177187-A1 DI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS Aventis Pharma Deutschland GmbH (DE) 2002-02-06 EP disclosed
WO-2000064888-A1 DI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-11-02 WO disclosed