SCHEMBL4842459

SCHEMBL4842459

COc1cc(NS(=O)(=O)c2cccc(Cl)c2)c(-c2ncno2)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
PKM P14618 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
PGR P06401 2/20 0.46
TP53 P04637 1/20 0.46
KDM1A O60341 1/20 0.46
PTGES2 Q9H7Z7 1/20 0.46
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
ALOX12 P18054 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CCR4 P51679 1/20 0.44
EDNRB P24530 2/20 0.44
EDNRA P25101 2/20 0.44
SLC40A1 Q9NP59 1/20 0.44
MAPT P10636 1/20 0.42
CCR2 P41597 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780513 0.86 ALDH1A1 (0.52) ALDH1A1PKMTSHRTP53KMT2A
SCHEMBL4781581 0.85 AXL (0.49) CYP3A4TSHRPTGES2KMT2AMEN1
SCHEMBL3089179 0.84 SLC40A1 (0.46) ALDH1A1TSHRPGRPTGES2EDNRB
SCHEMBL4781223 0.82 EDNRB (0.48) ALDH1A1CYP1A2CYP3A4PKMTSHR
SCHEMBL4775751 0.81 SLC40A1 (0.44) CYP2C19PGRKDM1ACCR4EDNRB
SCHEMBL3095682 0.78 PIK3C2B (0.36) ALDH1A1PKMPGRKDM1AKMT2A
SCHEMBL4836640 0.72 EDNRA (0.46) ALDH1A1TSHRTP53KMT2AMEN1
SCHEMBL4793152 0.70 SLC40A1 (0.46) ALDH1A1TSHRTP53KMT2AMEN1
SCHEMBL4782048 0.70 PGR (0.54) ALDH1A1PKMPGRKDM1AKMT2A
SCHEMBL16501001 0.70 AXL (0.47) CYP3A4KMT2AMEN1SLC40A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008008374-A2 CCR2 INHIBITORS AND METHODS OF USE THEREOF CHEMOCENTRYX, INC. (US) 2008-01-17 WO claimed