SCHEMBL4854868

SCHEMBL4854868

CC(=O)c1ccc(OCCN(C)C)cc1N1CCN(C)CC1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOB P27338 14/20 0.46
HTR1A P08908 1/20 0.44
HTR1D P28221 1/20 0.44
HTR1B P28222 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MGLL Q99685 1/20 0.42
ABHD6 Q9BV23 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3688257 0.79 ALDH1A1 (0.51) HTR1AHTR1DHTR1BKDM4EALDH1A1
SCHEMBL6141581 0.78 HTR1A (0.44) HTR1AHTR1DHTR1BKDM4EALDH1A1
SCHEMBL4855833 0.74 MAOB (0.58) MAOBKDM4EALDH1A1
SCHEMBL14922281 0.74 HRH3 (0.57) KDM4EALDH1A1
SCHEMBL8614407 0.73 ROCK1 (0.54) KDM4EALDH1A1MGLLABHD6
SCHEMBL3690359 0.72 GAA (0.57) KDM4EALDH1A1
SCHEMBL14590673 0.71 NOTUM (0.64) KDM4EALDH1A1
SCHEMBL17324776 0.70 HRH3 (0.47)
SCHEMBL3683974 0.68 HSD11B1 (0.38) MAOBHTR1BKDM4EALDH1A1
SCHEMBL12853694 0.68 MGLL (0.56) KDM4EALDH1A1MGLLABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed