SCHEMBL4882259

SCHEMBL4882259

O=C(NCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)c1cn[nH]c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 2/20 0.59
ROCK2 O75116 2/20 0.53
ROCK1 Q13464 2/20 0.53
ALDH1A1 P00352 5/20 0.49
KDM4E B2RXH2 3/20 0.49
HPGD P15428 5/20 0.48
CYP1A2 P05177 3/20 0.48
CYP2D6 P10635 3/20 0.48
CYP2C19 P33261 3/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C9 P11712 1/20 0.48
P2RX1 P51575 1/20 0.48
TMPRSS4 Q9NRS4 1/20 0.48
MTOR P42345 1/20 0.47
TACR1 P25103 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
GAA P10253 3/20 0.46
PLA2G1B P04054 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4879066 0.87 ROCK2 (0.68) MLYCDROCK2ROCK1HPGDCYP1A2
SCHEMBL4882240 0.86 MAPK14 (0.59) MLYCDROCK2ROCK1MAPK14
SCHEMBL18741154 0.78 ROCK2 (0.54) ROCK2ROCK1
SCHEMBL18741074 0.75 L3MBTL1 (0.61) ROCK2ROCK1CYP1A2CYP2C19CYP3A4
SCHEMBL4879445 0.75 ROCK2 (0.60) ROCK2ROCK1HPGD
SCHEMBL17065962 0.74 MARK3 (0.42) ROCK2ALDH1A1
SCHEMBL506527 0.73 MLYCD (0.72) MLYCDALDH1A1KDM4EHPGDCYP1A2
SCHEMBL6253464 0.73 MLYCD (0.60) MLYCDALDH1A1KDM4EHPGDCYP1A2
SCHEMBL4883200 0.72 MAOB (0.62) ROCK2ROCK1ALDH1A1HPGDMEN1
SCHEMBL360181 0.72 ROCK2 (0.65) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080064690-A1 PYRAZOLE-AMIDES AND -SULFONAMIDES ICAGEN, INC. (US) 2008-03-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080064690-A1 PYRAZOLE-AMIDES AND -SULFONAMIDES SCN3A, TRPV3, HCN3 MLYCD 3862/4885ROCK2 4342/4885ROCK1 4527/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.