7-Prenyloxycoumarin

7-Prenyloxycoumarin

SCHEMBL4898255

CC(C)=CCOc1ccc2ccc(=O)oc2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 1.00
ALDH1A1 P00352 4/20 1.00
MTNR1A P48039 2/20 1.00
ALOX15 P16050 4/20 0.79
CYP3A4 P08684 3/20 0.79
HPGD P15428 3/20 0.79
MAPT P10636 3/20 0.79
NDUFS8 O00217 3/20 0.79
COXFA4 O00483 3/20 0.79
NDUFAB1 O14561 3/20 0.79
NDUFA1 O15239 3/20 0.79
NDUFS4 O43181 3/20 0.79
NDUFB5 O43674 3/20 0.79
NDUFB3 O43676 3/20 0.79
NDUFC1 O43677 3/20 0.79
NDUFA2 O43678 3/20 0.79
NDUFS5 O43920 3/20 0.79
NDUFS7 O75251 3/20 0.79
NDUFS2 O75306 3/20 0.79
NDUFS6 O75380 3/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17898116 0.90 KDM4E (0.82) KDM4EALDH1A1MTNR1AALOX15CYP3A4
Auraptene SCHEMBL2535034 0.89 ALOX15 (1.00) KDM4EALDH1A1MTNR1AALOX15CYP3A4
Auraptene SCHEMBL2535029 0.89 ALOX15 (1.00) KDM4EALDH1A1MTNR1AALOX15CYP3A4
SCHEMBL18265492 0.88 KDM4E (0.78) KDM4EALDH1A1MTNR1AALOX15CYP3A4
Umbelliprenin SCHEMBL26641528 0.88 ALOX15 (1.00) KDM4EALDH1A1MTNR1AALOX15CYP3A4
Umbelliprenin SCHEMBL18265478 0.88 ALOX15 (1.00) KDM4EALDH1A1MTNR1AALOX15CYP3A4
Umbelliprenin SCHEMBL28133292 0.88 ALOX15 (1.00) KDM4EALDH1A1MTNR1AALOX15CYP3A4
SCHEMBL29999425 0.83 NDUFS8 (0.83) KDM4EALDH1A1MTNR1AALOX15CYP3A4
SCHEMBL24700226 0.82 NDUFS8 (0.81) KDM4EALDH1A1MTNR1AALOX15CYP3A4
SCHEMBL4390495 0.82 CA12 (0.75) KDM4EALDH1A1MTNR1AALOX15CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016193220-A1 SKIN PIGMENTATION MODIFIERS TO DARKEN OR LIGHTEN THE SKIN AFFICHEM (FR) 2016-12-08 WO disclosed
US-8729279-B2 Agent for promoting osteoblast differentiation, pharmaceutical composition for promoting bone formation, and food for special dietary use containing auraptene analog as active ingredient ERINA CO., INC. (JP) 2014-05-20 US disclosed
US-8729279-B2 Agent for promoting osteoblast differentiation, pharmaceutical composition for promoting bone formation, and food for special dietary use containing auraptene analog as active ingredient ERINA CO., INC. (JP) 2014-05-20 US disclosed
EP-2001463-B1 A PHARMACEUTICAL COMPOSITION USEFUL AS ACETYL CHOLINESTERASE INHIBITORS COUNCIL SCIENT IND RES (IN) 2013-07-03 EP disclosed
US-20130102796-A1 AGENT FOR PROMOTING OSTEOBLAST DIFFERENTIATION, PHARMACEUTICAL COMPOSITION FOR PROMOTING BONE FORMATION, AND FOOD FOR SPECIAL DIETARY USE CONTAINING AURAPTENE ANALOG AS ACTIVE INGREDIENT ERINA CO., INC. (JP) 2013-04-25 US disclosed
US-20130102796-A1 AGENT FOR PROMOTING OSTEOBLAST DIFFERENTIATION, PHARMACEUTICAL COMPOSITION FOR PROMOTING BONE FORMATION, AND FOOD FOR SPECIAL DIETARY USE CONTAINING AURAPTENE ANALOG AS ACTIVE INGREDIENT ERINA CO., INC. (JP) 2013-04-25 US disclosed
US-20120277297-A1 Pharmaceutical Composition Useful as Acetylcholinesterase Inhibitors COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2012-11-01 US disclosed
US-8188143-B2 Pharmaceutical composition useful as acetylcholinesterase inhibitors COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2012-05-29 US disclosed
US-20080009544-A1 Pharmaceutical Composition Useful as Acetylcholinesterase Inhibitors COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2008-01-10 US disclosed
WO-2003028762-A1 NOVEL ANTIMICROBIAL RESISTANCE BLOCKING COMPOSITIONS ETHICON, INC. (US) 2003-04-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080009544-A1 Pharmaceutical Composition Useful as Acetylcholinesterase Inhibitors ACHE, BCHE, CHRNB1 KDM4E 1482/4885ALDH1A1 1025/4885MTNR1A 302/4885
US-20130102796-A1 AGENT FOR PROMOTING OSTEOBLAST DIFFERENTIATION, PHARMACEUTICAL COMPOSITION FOR PROMOTING BONE FORMATION, AND FOOD FOR SPECIAL DIETARY USE CONTAINING AURAPTENE ANALOG AS ACTIVE INGREDIENT MYADM, EBP, HGFAC KDM4E 573/4885ALDH1A1 368/4885MTNR1A 390/4885
US-20120277297-A1 Pharmaceutical Composition Useful as Acetylcholinesterase Inhibitors ACHE, BCHE, CYP3A7 KDM4E 1461/4885ALDH1A1 547/4885MTNR1A 1278/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.