SCHEMBL4915938

SCHEMBL4915938

COC(=O)c1ccc2c(c1)[nH]c(=O)n2CCC(C)(C)NC(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.47
KDM4E B2RXH2 8/20 0.47
GAA P10253 8/20 0.47
HPGD P15428 5/20 0.47
KMT2A Q03164 4/20 0.47
GLA P06280 4/20 0.47
HSD17B10 Q99714 3/20 0.47
HTT P42858 2/20 0.47
PKM P14618 2/20 0.47
MEN1 O00255 3/20 0.43
RAB9A P51151 3/20 0.43
TDP1 Q9NUW8 1/20 0.40
EPHX2 P34913 1/20 0.40
MAPT P10636 3/20 0.39
PPARG P37231 1/20 0.38
NCOA2 Q15596 1/20 0.38
NCOA1 Q15788 1/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4640997 0.84 MEN1 (0.36) HPGDKMT2AMEN1RAB9AEPHX2
SCHEMBL4915808 0.83 KDM4E (0.53) ALDH1A1KDM4EGAAHPGDKMT2A
SCHEMBL5320024 0.79 ALDH1A1 (0.58) ALDH1A1KDM4EGAAHPGDKMT2A
SCHEMBL891359 0.77 KDM4E (0.47) ALDH1A1KDM4EGAAHPGDKMT2A
SCHEMBL9725397 0.76 ALDH1A1 (0.55) ALDH1A1KDM4EGAAHPGDKMT2A
SCHEMBL14530088 0.75 ALDH1A1 (0.54) ALDH1A1KDM4EGAAHPGDKMT2A
Hydrochloric Acid SCHEMBL9725495 0.75 ALDH1A1 (0.54) ALDH1A1KDM4EGAAHPGDKMT2A
SCHEMBL7214732 0.74 PARP1 (0.45) ALDH1A1KDM4EGAAHPGDKMT2A
SCHEMBL15183122 0.74 CNR2 (0.48) ALDH1A1KDM4EGAAHPGDKMT2A
SCHEMBL15687345 0.72 SMN1; SMN2 (0.58) ALDH1A1KDM4EGAAHPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080103138-A1 Beta-agonists, methods for the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-05-01 US disclosed
US-20080103138-A1 Beta-agonists, methods for the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-05-01 US disclosed
US-20080103138-A1 Beta-agonists, methods for the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-05-01 US disclosed
US-20070112033-A1 N-(3-{2-[3-(6-amino-benzimidazol-1-yl)-1,1-dimethyl-propylamino]-1-hydroxy-ethyl}-phenyl)-benzenesulphonamide; beta(3)-Adrenoceptor agonists; antidiabetic, obesity, insulin resistance BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-17 US disclosed
US-20070112033-A1 N-(3-{2-[3-(6-amino-benzimidazol-1-yl)-1,1-dimethyl-propylamino]-1-hydroxy-ethyl}-phenyl)-benzenesulphonamide; beta(3)-Adrenoceptor agonists; antidiabetic, obesity, insulin resistance BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-17 US disclosed
US-20070112033-A1 N-(3-{2-[3-(6-amino-benzimidazol-1-yl)-1,1-dimethyl-propylamino]-1-hydroxy-ethyl}-phenyl)-benzenesulphonamide; beta(3)-Adrenoceptor agonists; antidiabetic, obesity, insulin resistance BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080103138-A1 Beta-agonists, methods for the preparation thereof and their use as pharmaceutical compositions ADRB1, ADRB3, ADRB2 ALDH1A1 717/4885KDM4E 4614/4885GAA 1816/4885
US-20070112033-A1 N-(3-{2-[3-(6-amino-benzimidazol-1-yl)-1,1-dimethyl-propylamino]-1-hydroxy-ethyl}-phenyl)-benzenesulphonamide; beta(3)-Adrenoceptor agonists; antidiabetic, obesity, insulin resistance ADRB3, ADRB1, ADRA1B ALDH1A1 573/4885KDM4E 4097/4885GAA 1475/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.