SCHEMBL493471

SCHEMBL493471

CN(C)C(c1ccccc1)C1CCC(NC(=O)CCNC(=O)c2nc(-c3ccccn3)no2)CC1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRCP P42785 11/20 0.44
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
FAAH O00519 1/20 0.40
CES1 P23141 1/20 0.40
NCEH1 Q6PIU2 1/20 0.40
DAGLA Q9Y4D2 1/20 0.40
SMYD3 Q9H7B4 1/20 0.39
TSHR P16473 2/20 0.38
GABRA5 P31644 1/20 0.37
CYP3A4 P08684 1/20 0.37
EPHX2 P34913 1/20 0.37
KCNH2 Q12809 1/20 0.37
CACNA1C Q13936 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL494528 0.85 SMN1; SMN2 (0.39) NPC1RAB9ASMYD3TSHRKDM4E
SCHEMBL493504 0.85 SMN1; SMN2 (0.53) NPC1RAB9ADAGLAKDM4E
SCHEMBL493429 0.84 HPGD (0.51) KDM4E
SCHEMBL493213 0.83 KMT2A (0.41) NPC1RAB9ASMYD3
SCHEMBL493611 0.82 SMYD3 (0.43) NPC1RAB9ASMYD3TSHR
SCHEMBL493060 0.78 FAAH (0.44) PRCPNPC1RAB9AFAAHCES1
SCHEMBL493600 0.78 GHSR (0.40) NPC1RAB9AKDM4E
SCHEMBL493820 0.77 RAB9A (0.40) NPC1RAB9ATSHR
SCHEMBL492913 0.77 RAB9A (0.39) NPC1RAB9AKDM4E
SCHEMBL494415 0.77 TSHR (0.42) NPC1RAB9ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106055-B2 Substituted amide compounds GRUENENTHAL GMBH (DE) 2012-01-31 US claimed