SCHEMBL4970801

SCHEMBL4970801

CCNc1cc(-c2cc(F)c(F)c(C)c2F)nc(C#N)c1N

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.33
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
RECQL P46063 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3108861 0.70 PGK1 (0.41) CTSSALDH1A1HPGD
SCHEMBL27762078 0.70 LMNA (0.43) CTSSALDH1A1HPGD
SCHEMBL3114802 0.68 CTSK (0.55) CTSS
SCHEMBL4593268 0.65 CYP11B1 (0.38) CTSSSMN1; SMN2
SCHEMBL5022259 0.62 CTSK (0.48) CTSS
SCHEMBL4593579 0.60 REN (0.36) ALDH1A1
SCHEMBL27823325 0.60 CYP3A4 (0.41) ALDH1A1HPGDRECQL
SCHEMBL20226521 0.59 KDM4E (0.36) ALDH1A1HPGDRECQL
SCHEMBL30971084 0.59 MAPK8 (0.47) ALDH1A1HPGDSMN1; SMN2
SCHEMBL27895277 0.58 ALDH1A1 (0.40) ALDH1A1HPGDRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979351-A1 6-PHENYL-1H-IMIDAZO[4, 5-C]PYRIDINE-4-CARBONITRILE DERIVATIVES AS CATHEPSIN K AND S INHIBITORS N.V. Organon (NL) 2008-10-15 EP disclosed
WO-2007080191-A1 6-PHENYL-1H-IMIDAZO[4, 5-C]PYRIDINE-4-CARBONITRILE DERIVATIVES AS CATHEPSIN K AND S INHIBITORS N.V. ORGANON (NL) 2007-07-19 WO disclosed