Beclobrate

Beclobrate

SCHEMBL49779

CCOC(=O)C(C)(CC)Oc1ccc(Cc2ccc(Cl)cc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 1.00
PPARA Q07869 7/20 0.63
CYP1A2 P05177 3/20 0.63
CYP3A4 P08684 3/20 0.63
ABCB11 O95342 2/20 0.63
TSHR P16473 2/20 0.63
HTR2A P28223 2/20 0.63
PMP22 Q01453 2/20 0.63
PPARG P37231 5/20 0.49
ALDH1A1 P00352 3/20 0.47
MAPT P10636 4/20 0.44
MEN1 O00255 2/20 0.44
CYP2C19 P33261 2/20 0.44
KMT2A Q03164 2/20 0.44
ELANE P08246 2/20 0.44
CYP2D6 P10635 1/20 0.44
FABP2 P12104 2/20 0.43
SLC22A12 Q96S37 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
LMNA P02545 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Beclobrate SCHEMBL3950803 1.00 OPRK1 (1.00) OPRK1PPARACYP1A2CYP3A4ABCB11
SCHEMBL1935420 0.93 OPRK1 (0.86) OPRK1PPARACYP1A2CYP3A4ABCB11
SCHEMBL11071767 0.90 OPRK1 (0.81) OPRK1PPARACYP1A2CYP3A4ABCB11
SCHEMBL11063131 0.90 OPRK1 (0.81) OPRK1PPARACYP1A2CYP3A4ABCB11
SCHEMBL11070815 0.88 OPRK1 (0.79) OPRK1PPARACYP1A2CYP3A4ABCB11
SCHEMBL11470655 0.88 OPRK1 (0.79) OPRK1PPARACYP1A2CYP3A4ABCB11
SCHEMBL11068228 0.88 OPRK1 (0.78) OPRK1PPARACYP1A2CYP3A4ABCB11
SCHEMBL11072228 0.88 OPRK1 (0.78) OPRK1PPARACYP1A2CYP3A4ABCB11
SCHEMBL5997445 0.88 OPRK1 (0.78) OPRK1PPARACYP1A2CYP3A4ABCB11
SCHEMBL11074765 0.87 OPRK1 (0.76) OPRK1PPARACYP1A2CYP3A4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1601 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104523608-B A kind of hydrophilic amide suitable for dewatering medicament is birdsed of the same feather flock together compound self assembly particulate medicine-releasing system and preparation method thereof 张建祥 2018-04-24 CN claimed
EP-2649989-B1 Method for preparing a solid dispersion, solid dispersion obtained thereby and use thereof UNIV KING SAUD (SA) 2017-10-18 EP claimed
EP-2251038-B1 SOLID DISPERSION, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND PROCESSES FOR THE PRODUCTION OF BOTH ASKA PHARM CO LTD (JP) 2017-05-10 EP claimed
US-20160367645-A1 LYSOSOMAL ACID LIPASE THERAPY FOR NAFLD AND RELATED DISEASES CHILDREN'S HOSPITAL MEDICAL CENTER (US) 2016-12-22 US claimed
US-20150352094-A1 USE OF FATTY ACID NIACIN CONJUGATES FOR TREATING DISEASES CATABASIS PHARMACEUTICALS, INC. 2015-12-10 US claimed
EP-2941252-A2 USE OF FATTY ACID NIACIN CONJUGATES FOR TREATING DISEASES Catabasis Pharmaceuticals, Inc. (US) 2015-11-11 EP claimed
CN-104840963-A Medicine composition containing lipoprotein-associated phospholipase A2 inhibitors and application thereof HEBEI DONGKANG BIOTECHNOLOGY CO LTD 2015-08-19 CN claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
CN-104523608-A Hydrophilic amide polymer self-assembly particle drug release system suitable for hydrophobic drugs and preparation method thereof ZHANG JIANXIANG 2015-04-22 CN claimed
WO-2014107730-A2 USE OF FATTY ACID NIACIN CONJUGATES FOR TREATING DISEASES CATABASIS PHARMACEUTICALS, INC. (US) 2014-07-10 WO claimed
US-20020003179-A1 Media milling SKYEPHARMA AG (CH) 2002-01-10 US claimed
WO-2001085345-A1 MEDIA MILLING RTP PHARMA INC. (US) 2001-11-15 WO claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
US-6211206-B1 Pharmaceutical composition TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US claimed
US-6211207-B1 ANTIDIABETIC AGENTS AND INSULIN SENSITIVITY ENHANCER TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
US-6133293-A INSULIN SENSITIVITY ENHANCER IN COMBINATION WITH OTHER ANTIDIABETICS DIFFERING FROM THE ENHANCER IN THE MECHANISM OF ACTION; POTENT DEPRESSIVE EFFECT ON DIABETIC HYPERGLYCEMIA; 2,4-THIAZOLIDINEDIONES AND OXAZOLIDINEDIONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-10-17 US claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
WO-1998031360-A1 PHARMACEUTICAL COMPOSITION HAVING HIGH BIOAVAILABILITY AND METHOD FOR PREPARING IT PHARMA PASS (FR) 1998-07-23 WO claimed
US-4483999-A Phenoxy alkanoic acid derivatives having the ability to lower the level of fatty substances in the blood SIEGFRIED AKTIENGESELLSCHAFT (CH) 1984-11-20 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150352094-A1 USE OF FATTY ACID NIACIN CONJUGATES FOR TREATING DISEASES NAMPT, NNT, FASN OPRK1 3802/4885PPARA 112/4885CYP1A2 720/4885
US-20160367645-A1 LYSOSOMAL ACID LIPASE THERAPY FOR NAFLD AND RELATED DISEASES LIPC, PNLIP, LIPA OPRK1 4501/4885PPARA 275/4885CYP1A2 2710/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.