SCHEMBL5013459

SCHEMBL5013459

Oc1nc2c(N3CCN(CCc4ccccc4)CC3)cccc2s1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.52
ALDH1A1 P00352 1/20 0.52
KMT2A Q03164 1/20 0.52
CYP2C9 P11712 1/20 0.52
ADRA1D P25100 2/20 0.49
ADRA1A P35348 2/20 0.49
ADRA1B P35368 2/20 0.49
HTR1A P08908 3/20 0.48
DRD2 P14416 2/20 0.48
HTR2A P28223 1/20 0.45
CASP1 P29466 1/20 0.44
CASP4 P49662 1/20 0.44
CASP5 P51878 1/20 0.44
HTR2C P28335 1/20 0.44
BCHE P06276 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5015080 0.77 DRD2 (0.41) MEN1ALDH1A1KMT2ADRD2
SCHEMBL5016133 0.77 KMT2A (0.51) MEN1ALDH1A1KMT2ACASP1BCHE
SCHEMBL5011693 0.73 ADRA1A (0.45) ALDH1A1CYP2C9ADRA1DADRA1AADRA1B
SCHEMBL8544808 0.73 MEN1 (0.51) MEN1ALDH1A1KMT2ACYP2C9ADRA1D
Hydrochloric Acid SCHEMBL8591257 0.73 MEN1 (0.51) MEN1ALDH1A1KMT2ACYP2C9ADRA1D
Hydrochloric Acid SCHEMBL6017322 0.72 CYP2C9 (0.50) MEN1ALDH1A1KMT2ACYP2C9ADRA1D
SCHEMBL8687612 0.71 HTR6 (0.61) MEN1ALDH1A1KMT2ACYP2C9ADRA1D
Hydrochloric Acid SCHEMBL9212305 0.71 CYP2C9 (0.49) MEN1ALDH1A1KMT2ACYP2C9ADRA1D
SCHEMBL5011767 0.71 HRH3 (0.45) CYP2C9ADRA1DADRA1AADRA1BHTR1A
SCHEMBL8549877 0.71 HTR1A (0.54) MEN1ALDH1A1KMT2ACYP2C9ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-B1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMA CO LTD (JP) 2008-10-08 EP disclosed