SCHEMBL5016131

SCHEMBL5016131

[O]c1nc2c(N3CCN(Cc4ccccc4F)CC3)cccc2s1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.51
KMT2A Q03164 5/20 0.51
KDM4E B2RXH2 3/20 0.51
POLB P06746 2/20 0.49
BCHE P06276 1/20 0.48
ACHE P22303 1/20 0.48
TSHR P16473 1/20 0.46
LMNA P02545 1/20 0.44
GNRHR P30968 1/20 0.43
ALDH3A1 P30838 1/20 0.43
HTR7 P34969 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MEN1 O00255 3/20 0.42
ATM Q13315 1/20 0.42
CYP2A13 Q16696 1/20 0.42
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
DRD4 P21917 2/20 0.42
DRD3 P35462 1/20 0.42
CASP1 P29466 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5016133 0.86 KMT2A (0.51) ALDH1A1KMT2AKDM4EPOLBBCHE
SCHEMBL5015107 0.84 GNRHR (0.44) ALDH1A1KMT2AKDM4EPOLBBCHE
SCHEMBL5013346 0.84 KDM4E (0.45) ALDH1A1KMT2AKDM4EPOLBBCHE
SCHEMBL2090166 0.82 DRD2 (0.40) KMT2APOLBBCHEACHETSHR
SCHEMBL27644481 0.78 ALDH1A1 (0.52) ALDH1A1KMT2AKDM4EPOLBTSHR
SCHEMBL5015079 0.77 DRD2 (0.41) KMT2ALMNANPSR1MEN1RAB9A
SCHEMBL27666519 0.76 POLB (0.64) ALDH1A1KMT2AKDM4EPOLBTSHR
SCHEMBL2093651 0.73 SCD (0.44) TSHRRAB9ANPC1
SCHEMBL5016197 0.72 DRD2 (0.43) ALDH1A1KMT2AKDM4ETSHRLMNA
SCHEMBL5011693 0.72 ADRA1A (0.45) ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-B1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMA CO LTD (JP) 2008-10-08 EP disclosed