SCHEMBL5047987

SCHEMBL5047987

CCCCCCCCCCCCNC(=O)c1cc(Br)c(CC(NC(=O)C(=O)O)c2cccc(-c3ccc(F)cc3)c2)c(Br)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.41
NAAA Q02083 1/20 0.40
DRD2 P14416 2/20 0.39
DRD4 P21917 2/20 0.39
DRD3 P35462 2/20 0.39
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
ASAH1 Q13510 1/20 0.38
LMNA P02545 2/20 0.38
TP53 P04637 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
HIF1A Q16665 1/20 0.38
ALOX15 P16050 2/20 0.36
MEN1 O00255 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5048336 0.85 NAAA (0.41) PTGS2NAAADRD2DRD4DRD3
SCHEMBL6022121 0.83 GPR139 (0.43) PTGS2NAAAHDAC1HDAC2LMNA
SCHEMBL6022152 0.76 DRD2 (0.43) NAAADRD2DRD4DRD3ASAH1
SCHEMBL6022126 0.76 ALDH1A1 (0.46) NAAAHDAC1HDAC2LMNASMN1; SMN2
SCHEMBL1854176 0.76 NAAA (0.40) NAAADRD2DRD4DRD3HDAC1
SCHEMBL5043892 0.75 GLI1 (0.43) HDAC1HDAC2NPC1RAB9AHIF1A
SCHEMBL6022090 0.75 GLI1 (0.43) HDAC1HDAC2NPC1RAB9AHIF1A
SCHEMBL5047944 0.73 DRD2 (0.46) PTGS2NAAADRD2DRD4DRD3
SCHEMBL5047162 0.73 HDAC1 (0.44) PTGS2NAAADRD2DRD4DRD3
SCHEMBL5039660 0.73 HDAC1 (0.44) PTGS2NAAADRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732534-B1 USE OF METHYLENE AMIDE DERIVATIVES IN CARDIOVASCULAR DISORDERS SERONO LAB (CH) 2008-07-23 EP disclosed