SCHEMBL5082292

SCHEMBL5082292

CC[C@H](N[C@H](C)c1ccccc1)C(=O)c1ccccc1.CS(=O)(=O)O

nearest known ligand 0.56

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRA2A known ✓ P08913 1/20 0.42
ADRA2B known ✓ P18089 1/20 0.42
HTR2A known ✓ P28223 1/20 0.42
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
LMNA P02545 1/20 0.46
HSD17B10 Q99714 1/20 0.46
APAF1 O14727 1/20 0.44
GPR139 Q6DWJ6 2/20 0.43
PGR P06401 1/20 0.42
HRH1 P35367 1/20 0.42
KCNH2 Q12809 1/20 0.42
ALDH1A1 P00352 2/20 0.42
MMP2 P08253 2/20 0.41
MMP9 P14780 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5079891 0.94 MEN1 (0.51) MEN1KMT2ALMNAHSD17B10APAF1
SCHEMBL5082805 0.82 ACP3 (0.47) KMT2ALMNAHSD17B10GPR139ALDH1A1
SCHEMBL652495 0.80 MEN1 (0.56) MEN1KMT2ALMNAHSD17B10APAF1
SCHEMBL17161710 0.77 MEN1 (0.53) MEN1KMT2AAPAF1ALDH1A1
SCHEMBL5082435 0.75 ACP3 (0.53) LMNAHSD17B10GPR139ALDH1A1TDP1
SCHEMBL22828969 0.75 ACP3 (0.53) LMNAHSD17B10GPR139ALDH1A1TDP1
SCHEMBL29961075 0.75 MMP8 (0.51) MEN1KMT2ALMNAAPAF1ALDH1A1
Hydrochloric Acid SCHEMBL22828960 0.73 ACP3 (0.56) LMNAHSD17B10GPR139ALDH1A1TDP1
Hydrochloric Acid SCHEMBL22828987 0.73 ACP3 (0.56) LMNAHSD17B10GPR139ALDH1A1TDP1
SCHEMBL5082297 0.73 ALDH1A1 (0.45) MEN1KMT2ALMNAALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7408084-B2 Process for producing optically active β-amino alcohol KANEKA CORPORATION (JP) 2008-08-05 US disclosed
US-20050277791-A1 Process for producing optically active beta-amino alcohol KANEKA CORPORATION (JP) 2005-12-15 US disclosed
EP-1512677-A1 PROCESS FOR PRODUCING OPTICALLY ACTIVE s-AMINO ALCOHOL KANEKA CORPORATION (JP) 2005-03-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050277791-A1 Process for producing optically active beta-amino alcohol ADH1A, ALDH7A1, ADH1C ADRA2A 221/4885ADRA2B 141/4885HTR2A 2049/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.