SCHEMBL5082297

SCHEMBL5082297

CC[C@H](NCCc1ccccc1)C(=O)c1ccccc1.CS(=O)(=O)O

nearest known ligand 0.45

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.45
MAPT P10636 3/20 0.45
LMNA P02545 2/20 0.45
GAA P10253 2/20 0.45
KDM4E B2RXH2 1/20 0.45
CYP3A4 P08684 1/20 0.45
BLM P54132 1/20 0.45
GFER P55789 1/20 0.45
PMP22 Q01453 1/20 0.45
AKR1C3 P42330 1/20 0.45
POLB P06746 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.43
OPRK1 P41145 1/20 0.43
HDAC2 Q92769 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
SIGMAR1 Q99720 2/20 0.42
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5079892 0.94 POLB (0.49) ALDH1A1MAPTLMNAGAAPOLB
SCHEMBL5082809 0.83 KMT2A (0.48) ALDH1A1MAPTLMNAGAAKDM4E
SCHEMBL27849653 0.81 POLB (0.53) ALDH1A1MAPTCYP3A4POLBOPRK1
SCHEMBL27586127 0.79 KMT2A (0.54) LMNAPOLBKMT2ASIGMAR1TP53
SCHEMBL5082438 0.76 SIGMAR1 (0.53) ALDH1A1MAPTGAAL3MBTL1OPRK1
SCHEMBL5082292 0.73 MEN1 (0.47) ALDH1A1LMNACYP3A4L3MBTL1MEN1
SCHEMBL5082242 0.73 NPC1 (0.46) ALDH1A1MAPTGAAL3MBTL1MEN1
SCHEMBL5079098 0.72 NPC1 (0.43) ALDH1A1MAPTPOLBOPRK1MEN1
SCHEMBL28190506 0.72 LMNA (0.49) ALDH1A1MAPTLMNAKDM4ECYP3A4
SCHEMBL6321040 0.72 HAT1 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7408084-B2 Process for producing optically active β-amino alcohol KANEKA CORPORATION (JP) 2008-08-05 US disclosed
US-20050277791-A1 Process for producing optically active beta-amino alcohol KANEKA CORPORATION (JP) 2005-12-15 US disclosed
EP-1512677-A1 PROCESS FOR PRODUCING OPTICALLY ACTIVE s-AMINO ALCOHOL KANEKA CORPORATION (JP) 2005-03-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050277791-A1 Process for producing optically active beta-amino alcohol ADH1A, ALDH7A1, ADH1C ALDH1A1 93/4885MAPT 2117/4885LMNA 1549/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.