SCHEMBL5088924

SCHEMBL5088924

O=C(O)COC1CCN(S(=O)(=O)c2ccc(Cl)cc2)C1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.50
PKM P14618 2/20 0.49
USP5 P45974 1/20 0.48
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
CNR1 P21554 1/20 0.48
GAA P10253 1/20 0.47
PTGIR P43119 1/20 0.47
POLB P06746 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5131530 0.88 MEN1 (0.51) LMNAPKMUSP5ALDH1A1SMN1; SMN2
SCHEMBL5093752 0.88 MAPT (0.55) PKMUSP5ALDH1A1KDM4EKMT2A
SCHEMBL5122649 0.88 ALDH1A1 (0.54) LMNAUSP5ALDH1A1KDM4EMEN1
SCHEMBL5093760 0.83 TRPV4 (0.52) LMNAUSP5ALDH1A1KDM4ESMN1; SMN2
SCHEMBL494593 0.81 CNR1 (0.50) CNR1PTGIR
SCHEMBL5125471 0.81 CYP2C19 (0.57) LMNAALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL5131953 0.80 MEN1 (0.56) LMNAPKMUSP5ALDH1A1SMN1; SMN2
SCHEMBL5085809 0.80 TSHR (0.54) SMN1; SMN2MEN1KMT2AGAAPOLB
SCHEMBL5121390 0.78 PKLR (0.49) LMNAPKMALDH1A1SMN1; SMN2MEN1
SCHEMBL5915284 0.77 LMNA (0.62) LMNAPKMALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8580965-B2 Substituted sulfonamide compounds GRUENENTHAL GMBH (DE) 2013-11-12 US disclosed
US-8580965-B2 Substituted sulfonamide compounds GRUENENTHAL GMBH (DE) 2013-11-12 US disclosed
US-8580965-B2 Substituted sulfonamide compounds GRUENENTHAL GMBH (DE) 2013-11-12 US disclosed
US-20080306084-A1 Substituted Amide Compounds GRUENENTHAL GMBH (DE) 2008-12-11 US disclosed
US-20080249128-A1 Substituted Sulfonamide Compounds GRUENENTHAL GMBH (DE) 2008-10-09 US disclosed
US-20080249128-A1 Substituted Sulfonamide Compounds GRUENENTHAL GMBH (DE) 2008-10-09 US disclosed
US-20080249128-A1 Substituted Sulfonamide Compounds GRUENENTHAL GMBH (DE) 2008-10-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080249128-A1 Substituted Sulfonamide Compounds BDKRB1, BDKRB2, NPSR1 LMNA 1324/4885PKM 1198/4885USP5 4128/4885
US-20080306084-A1 Substituted Amide Compounds OPRK1, NAA50, ACMSD LMNA 2485/4885PKM 1161/4885USP5 3994/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.