SCHEMBL5187264

SCHEMBL5187264

CN(Cc1ccccc1)C(=O)Oc1ccc(CN2CCCC2)n1C

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BCHE P06276 6/20 0.46
HTT P42858 2/20 0.43
PKM P14618 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HRH3 Q9Y5N1 3/20 0.43
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
CXCR4 P61073 2/20 0.42
ACHE P22303 5/20 0.42
KCNH2 Q12809 1/20 0.41
LMNA P02545 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CPT2 P23786 1/20 0.41
CPT1A P50416 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5187738 0.90 ACHE (0.47) BCHEHTTKDM4EALDH1A1ACHE
SCHEMBL5188684 0.85 KDM4E (0.45) BCHEKDM4EALDH1A1LMNAMEN1
SCHEMBL5189076 0.78 HTR1A (0.45) HTTSMN1; SMN2HRH3KDM4EALDH1A1
SCHEMBL4658971 0.73 HRH3 (0.64) BCHEHRH3CXCR4ACHE
SCHEMBL5188224 0.72 KDM4E (0.43) KDM4EALDH1A1LMNAMEN1KMT2A
SCHEMBL3762996 0.72 ACHE (0.49) BCHEHTTKDM4EALDH1A1ACHE
SCHEMBL5186000 0.71 NPC1 (0.47) SMN1; SMN2MEN1KMT2A
SCHEMBL31164812 0.68 NPC1 (0.61) SMN1; SMN2MEN1KMT2A
N-Benzylmethylamine SCHEMBL5556336 0.68 NCF1 (0.50) HRH3KDM4EKMT2A
SCHEMBL2095210 0.68 NPC1 (0.67) SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751101-B1 Substituted 5-aminomethyl-1H-pyrrole-2-carboxylic acid amides GRUENENTHAL GMBH (DE) 2012-11-14 EP claimed
EP-1751101-A1 SUBSTITUTED 5-AMINOMETHYL-1H-PYRROL-2-CARBXYLIC ACID AMIDES Grünenthal GmbH (DE) 2007-02-14 EP claimed
WO-2005113497-A1 SUBSTITUTED 5-AMINOMETHYL-1H-PYRROL-2-CARBXYLIC ACID AMIDES Grünenthal GmbH (DE) 2005-12-01 WO claimed