SCHEMBL5193335

SCHEMBL5193335

CCOc1ccc(CNC(=O)CC2CN(Cc3cccnc3)CCN2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.49
TP53 P04637 3/20 0.49
LMNA P02545 3/20 0.49
ALDH1A1 P00352 3/20 0.49
MAPK1 P28482 2/20 0.49
POLB P06746 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
KMT2A Q03164 2/20 0.47
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
KDM4E B2RXH2 2/20 0.46
TSHR P16473 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
LTA4H P09960 1/20 0.44
GAA P10253 1/20 0.43
NAMPT P43490 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5195331 0.91 GAA (0.49) SMN1; SMN2LMNAALDH1A1POLBKMT2A
SCHEMBL5190900 0.82 POLB (0.49) ALDH1A1POLBTDP1KMT2ANPC1
SCHEMBL5192049 0.77 KDM4E (0.43) SMN1; SMN2POLBKMT2AKDM4ENPC1
SCHEMBL5191569 0.76 ALDH1A1 (0.47) ALDH1A1MAPK1TDP1KMT2AKDM4E
SCHEMBL5192336 0.75 ALDH1A1 (0.51) ALDH1A1TDP1KMT2ARAB9AGAA
SCHEMBL5192704 0.73 NOS2 (0.56)
SCHEMBL5193118 0.72 NOS2 (0.57)
SCHEMBL5193328 0.71 L3MBTL1 (0.49) SMN1; SMN2LMNAALDH1A1MAPK1POLB
SCHEMBL5193835 0.71 ALDH1A1 (0.48) SMN1; SMN2ALDH1A1KMT2ACYP3A4CYP2C9
SCHEMBL13535271 0.70 KMT2A (0.49) ALDH1A1MAPK1POLBTDP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed