SCHEMBL5205016

SCHEMBL5205016

S=C1Nc2ccc(Cl)cc2C(c2ccccc2)N1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
ALOX12 P18054 1/20 0.44
ATM Q13315 1/20 0.43
KIF11 P52732 1/20 0.43
KMT2A Q03164 6/20 0.43
MEN1 O00255 5/20 0.43
GAA P10253 3/20 0.42
TRPM5 Q9NZQ8 3/20 0.41
TRPM4 Q8TD43 2/20 0.41
MAPT P10636 3/20 0.40
KDM4E B2RXH2 1/20 0.40
GLA P06280 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5177579 0.88 ALDH1A1 (0.46) ALDH1A1ALOX12KIF11KMT2AMEN1
SCHEMBL5696173 0.85 DHFR (0.50) ALDH1A1ALOX12ATMKIF11KMT2A
SCHEMBL5177430 0.84 MAPT (0.50) ALDH1A1ALOX12ATMKMT2AMEN1
SCHEMBL5177359 0.82 ALDH1A1 (0.54) ALDH1A1ATMKIF11KMT2AMEN1
SCHEMBL13612701 0.82 ALDH1A1 (0.46) ALDH1A1KMT2AMEN1GAAMAPT
SCHEMBL5178013 0.81 KMT2A (0.55) ALDH1A1ALOX12KMT2AMEN1GAA
SCHEMBL5696272 0.81 CHRM1 (0.42) ALDH1A1ALOX12KMT2AGAAMAPT
SCHEMBL9567855 0.80 ALDH1A1 (0.54) ALDH1A1KMT2AMEN1GAAMAPT
SCHEMBL5176626 0.80 ALDH1A1 (0.54) ALDH1A1KMT2AMEN1GAAMAPT
SCHEMBL5696249 0.74 DHFR (0.51) ALDH1A1KIF11TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807402-A1 QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION, THEIR USE AS ANTIMITOTICS AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAID DERIVATIVES EMBL (DE) 2007-07-18 EP disclosed
WO-2006048308-A1 QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION, THEIR USE AS ANTIMITOTICS AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAID DERIVATIVES EMBL (DE) 2006-05-11 WO disclosed
EP-1655289-A1 Quinazoline derivatives, process for their preparation, their use as antimitotics and pharmaceutical compositions comprising said derivatives EMBL (DE) 2006-05-10 EP disclosed
EP-0564397-A1 Antiatherosclerotic substituted phenylquinazoline derivatives SANDOZ LTD. (CH) 1993-10-06 EP disclosed