SCHEMBL5696272

SCHEMBL5696272

Fc1ccccc1C1NC(=S)Nc2ccc(Cl)cc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 7/20 0.42
GAA P10253 5/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HTT P42858 1/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
TDP1 Q9NUW8 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MAPT P10636 3/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
CASP1 P29466 1/20 0.40
CYP2C19 P33261 1/20 0.40
RECQL P46063 1/20 0.40
SLC8B1 Q6J4K2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5177430 0.86 MAPT (0.50) GAAALDH1A1HTR2AHTR2CTDP1
SCHEMBL5176914 0.83 LMNA (0.41) GAAALDH1A1LMNAKDM4EHTT
SCHEMBL5205016 0.81 ALDH1A1 (0.46) CHRM1GAAALDH1A1KDM4EMAPT
SCHEMBL10925308 0.75 CHRM1 (0.45) CHRM1GAAALDH1A1LMNAHTT
SCHEMBL23721282 0.74 LMNA (0.42) GAALMNAHTR2AHTR2CMAPT
SCHEMBL5696173 0.73 DHFR (0.50) ALDH1A1HTTHTR2AHTR2CMAPT
SCHEMBL5178013 0.72 KMT2A (0.55) GAAALDH1A1LMNAKDM4EHTT
SCHEMBL4590461 0.71 CACNB4 (0.47) LMNAMAPTTP53CYP1A2CYP2C9
SCHEMBL11083785 0.70 CHRM1 (0.41) CHRM1GAAALDH1A1LMNAHTT
SCHEMBL7313268 0.70 HTR2C (0.39) CHRM1GAAHTR2AHTR2CMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1655289-A1 Quinazoline derivatives, process for their preparation, their use as antimitotics and pharmaceutical compositions comprising said derivatives EMBL (DE) 2006-05-10 EP disclosed