SCHEMBL5487349

SCHEMBL5487349

CN(C)C(=O)Cn1cc(C2CCN(S(=O)(=O)Cc3ccccc3)C2)c2ccccc21.Cc1ccc(F)c(C(=O)N2CCC(c3cn(Cc4ccc(C#N)cc4)c4ccccc34)C2)c1Cl.Cc1ccc(S(=O)(=O)NC(Cc2ccccc2)C(=O)N2CCC(c3cn(CC(=O)N(C)C)c4ccccc34)C2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 7/20 0.36
HPN P05981 2/20 0.36
ST14 Q9Y5Y6 2/20 0.36
HGFAC Q04756 1/20 0.36
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
F11 P03951 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HTR6 P50406 1/20 0.33
ATM Q13315 1/20 0.33
SMO Q99835 1/20 0.32
P2RX7 Q99572 1/20 0.32
MMP2 P08253 1/20 0.32
MMP13 P45452 1/20 0.32
MMP14 P50281 1/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
THRB P10828 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5202889 0.80 HPN (0.52) ADAM17HPNST14HGFACKMT2A
SCHEMBL5205062 0.78 SMO (0.46) ALDH1A1SMOLMNAPOLBHTT
SCHEMBL5203062 0.71 HCRTR1 (0.49) ALDH1A1HTR6LMNAPOLBTHRB
SCHEMBL4860552 0.67 HRH2 (0.46) KMT2AALDH1A1LMNA
SCHEMBL5822858 0.65 HRH2 (0.35) SMO
SCHEMBL5202142 0.65 LMNA (0.50) ALDH1A1HTR6SMOLMNAPOLB
SCHEMBL5206068 0.64 LMNA (0.49) ALDH1A1HTR6SMOLMNAPOLB
SCHEMBL4859112 0.64 RORC (0.47) ALDH1A1HTR6LMNAPOLB
SCHEMBL4854486 0.63 ALDH1A1 (0.46) KMT2AALDH1A1MEN1KDM4E
SCHEMBL4851493 0.63 MEN1 (0.45) KMT2AMEN1HTR6ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007501828-A 2007-02-01 JP claimed
EP-1654253-A1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES Grünenthal GmbH (DE) 2006-05-10 EP claimed
WO-2005019208-A1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES Grünenthal GmbH (DE) 2005-03-03 WO claimed