SCHEMBL5210504

SCHEMBL5210504

Cc1ccc(C(=O)O)c(NC(=O)Cc2c[nH]c3ccc(F)cc23)c1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.56
ANO1 Q5XXA6 1/20 0.51
MPO P05164 7/20 0.48
NOTUM Q6P988 2/20 0.47
MTNR1A P48039 2/20 0.47
MTNR1B P49286 2/20 0.47
KDM4E B2RXH2 1/20 0.47
SPR P35270 1/20 0.46
MAPT P10636 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
GPR84 Q9NQS5 1/20 0.44
SLC6A4 P31645 1/20 0.44
ICMT O60725 1/20 0.43
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5206707 0.92 ICMT (0.53) TSHRANO1MPOMTNR1AMTNR1B
SCHEMBL5209045 0.87 CDK2 (0.49) MTNR1AMTNR1BMAPTNPSR1GPR84
SCHEMBL5210851 0.86 MAPT (0.60) TSHRMAPTNPSR1POLBSMN1; SMN2
SCHEMBL5207887 0.85 KDM4E (0.60) MPONOTUMMTNR1AMTNR1BKDM4E
SCHEMBL5213599 0.81 ICMT (0.61) KDM4EMAPTNPSR1ICMT
SCHEMBL5211211 0.81 HTR1D (0.48) MAPTNPSR1ICMTPOLBSMN1; SMN2
SCHEMBL5214070 0.81 PPARG (0.57) KDM4EMAPTSLC6A4POLBSMN1; SMN2
SCHEMBL5213952 0.81 ICMT (0.47) KDM4EMAPTNPSR1ICMTSMN1; SMN2
SCHEMBL5207800 0.80 ICMT (0.51) MTNR1AMTNR1BKDM4EICMT
SCHEMBL5208637 0.79 ICMT (0.49) MAPTICMTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7288564-B2 Indole derivatives GLAXO GROUP LIMITED (GB) 2007-10-30 US claimed
US-7288564-B2 Indole derivatives GLAXO GROUP LIMITED (GB) 2007-10-30 US disclosed
EP-1343757-B1 INDOLE DERIVATIVES GLAXO GROUP LTD (GB) 2007-02-14 EP disclosed
US-20040092569-A1 Indole derivatives GLAXO GROUP LIMITED (GB) 2004-05-13 US disclosed
EP-1343757-A1 INDOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 2003-09-17 EP disclosed
WO-2002050031-A1 INDOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 2002-06-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040092569-A1 Indole derivatives PTGER4, PTGER1, TRPV4 TSHR 1260/4885ANO1 2417/4885MPO 4206/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.