SCHEMBL5211511

SCHEMBL5211511

CSCC[C@H](N)C(=O)OC(C)(C)C

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 2/20 0.43
NOS3 P29474 1/20 0.43
NOS2 P35228 1/20 0.43
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
RNPEP Q9H4A4 1/20 0.37
LTA4H P09960 1/20 0.37
METAP2 P50579 1/20 0.37
METAP1 P53582 1/20 0.37
MARS1 P56192 5/20 0.36
HSD17B10 Q99714 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ANPEP P15144 1/20 0.35
ENPEP Q07075 1/20 0.35
BHMT Q93088 3/20 0.35
CA2 P00918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11119448 1.00 NOS1 (0.43) NOS1NOS3NOS2CTSSCTSK
SCHEMBL7157725 1.00 NOS1 (0.43) NOS1NOS3NOS2CTSSCTSK
Hydrochloric Acid SCHEMBL918798 0.98 NOS1 (0.42) NOS1NOS3NOS2CTSSCTSK
Hydrochloric Acid SCHEMBL5211496 0.98 NOS1 (0.42) NOS1NOS3NOS2CTSSCTSK
SCHEMBL27863494 0.89 NOS1 (0.41) NOS1NOS3NOS2CTSSCTSK
SCHEMBL16618514 0.86 CTSS (0.38) NOS1NOS3NOS2CTSSCTSK
SCHEMBL3294154 0.84 NOS1 (0.42) NOS1NOS3NOS2CTSKLTA4H
SCHEMBL10683562 0.84 NOS1 (0.42) NOS1NOS3NOS2LTA4HMETAP2
SCHEMBL24786178 0.83 METAP2 (0.34) CTSSCTSKRNPEPMETAP2METAP1
SCHEMBL918772 0.82 NOS1 (0.43) NOS1NOS3NOS2CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 82 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1301660-C Method for supplying bioavailable methionine to cow AVENTIS ANIMAL NUTRITION SA (IE) 2007-02-28 CN claimed
CN-1326322-A Method for supplying bioavailable methionine to cow AVENTIS ANIMAL NUTRITION SA (FR) 2001-12-12 CN claimed
EP-4306530-B1 SILANE-CONTAINING CONDENSED CYCLIC DIPEPTIDE COMPOUND, PRODUCTION METHOD THEREFOR, AND METHOD FOR PRODUCING POLYPEPTIDE COMPOUND USING SAME CHUBU UNIV EDUCATIONAL FOUNDATION (JP) 2026-04-01 EP disclosed
US-20250375544-A1 DUAL MODE RADIOTRACER AND -THERAPEUTICS UNIV MUENCHEN TECH (DE) 2025-12-11 US disclosed
EP-4538279-A2 REACTION AGENT FOR AMIDE REACTIONS AND AMIDE COMPOUND PRODUCTION METHOD USING SAME Chubu University Educational Foundation (JP) 2025-04-16 EP disclosed
US-20240209020-A1 REACTION AGENT FOR AMIDE REACTION AND METHOD FOR PRODUCING AMIDE COMPOUND USING SAME CHUBU UNIVERSITY EDUCATIONAL FOUNDATION (JP) 2024-06-27 US disclosed
US-20240182517-A1 SILANE-CONTAINING CONDENSED CYCLIC DIPEPTIDE COMPOUND, PRODUCTION METHOD THEREFOR, AND METHOD FOR PRODUCING POLYPEPTIDE COMPOUND USING SAME CHUBU UNIVERSITY EDUCATIONAL FOUNDATION (JP) 2024-06-06 US disclosed
EP-4306530-A1 SILANE-CONTAINING CONDENSED CYCLIC DIPEPTIDE COMPOUND, PRODUCTION METHOD THEREFOR, AND METHOD FOR PRODUCING POLYPEPTIDE COMPOUND USING SAME Chubu University Educational Foundation (JP) 2024-01-17 EP disclosed
EP-4271422-A1 DUAL MODE RADIOTRACER AND -THERAPEUTICS Technische Universität München (DE) 2023-11-08 EP disclosed
CN-116981486-A Dual mode radiotracer and therapeutic agent 慕尼黑工业大学 2023-10-31 CN disclosed
EP-3334710-B1 COMPOSITIONS AND METHODS FOR TREATING AND PREVENTING NEURODEGENERATIVE DISORDERS ALZHEON INC (US) 2023-10-04 EP disclosed
WO-1998032741-A1 INHIBITORS OF FARNESYL PROTEIN TRANSFERASE ZENECA LIMITED (GB) 1998-07-30 WO disclosed
US-5786480-A ANTITUMOR AGENT; VIRICIDES SCHERING CORPORATION (US) 1998-07-28 US disclosed
WO-1998011073-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1998-03-19 WO disclosed
WO-1998007713-A1 HIGH MOLECULAR WEIGHT POLYMER-BASED PRODRUGS ENZON, INC. (US) 1998-02-26 WO disclosed
EP-0750609-A4 ISOPRENYL TRANSFERASE INHIBITORS EISAI CO LTD (JP) 1997-09-24 EP disclosed
US-5608067-A ANTITUMOR AGENTS MERCK SHARP & DOHME CORP. 1997-03-04 US disclosed
EP-0750609-A1 ISOPRENYL TRANSFERASE INHIBITORS Eisai Co., Ltd. (JP) 1997-01-02 EP disclosed
WO-1995025086-A1 ISOPRENYL TRANSFERASE INHIBITORS EISAI CO., LTD. (JP) 1995-09-21 WO disclosed
EP-0618221-A2 Heterocyclic inhibitors of farnesyl protein transferase BRISTOL-MYERS SQUIBB COMPANY (US) 1994-10-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250375544-A1 DUAL MODE RADIOTRACER AND -THERAPEUTICS MAN2B1, GBA1, SSTR1 NOS1 3459/4885NOS3 4753/4885NOS2 4741/4885
US-20240209020-A1 REACTION AGENT FOR AMIDE REACTION AND METHOD FOR PRODUCING AMIDE COMPOUND USING SAME NAAA, FAAH, FAAH2 NOS1 365/4885NOS3 1587/4885NOS2 626/4885
US-20240182517-A1 SILANE-CONTAINING CONDENSED CYCLIC DIPEPTIDE COMPOUND, PRODUCTION METHOD THEREFOR, AND METHOD FOR PRODUCING POLYPEPTIDE COMPOUND USING SAME VIP, NGLY1, NPR1 NOS1 186/4885NOS3 796/4885NOS2 262/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.