SCHEMBL5213651

SCHEMBL5213651

O=S(=O)(CCC[CH]C1CCNCC1)N1CCN(C2CCCC2)CC1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.37
KDM4E B2RXH2 5/20 0.37
HRH3 Q9Y5N1 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALOX15 P16050 1/20 0.35
MAPK1 P28482 2/20 0.33
HTR4 Q13639 1/20 0.33
HSD17B10 Q99714 1/20 0.32
POLB P06746 2/20 0.32
TP53 P04637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
GAA P10253 1/20 0.32
ITGB3 P05106 1/20 0.30
ITGA2B P08514 1/20 0.30
F2R P25116 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5213847 0.85 ALDH1A1 (0.31) ALDH1A1HTR4
SCHEMBL5219348 0.85 KDM4E (0.39) KDM4EITGB3ITGA2BF2R
SCHEMBL5216238 0.85 KDM4E (0.33) KDM4EKMT2AHTR4
SCHEMBL5212276 0.83 IKBKB (0.32) HTR4
SCHEMBL5215599 0.81 KDM4E (0.34) ALDH1A1KDM4EKMT2AHTR4
SCHEMBL5215923 0.80 LMNA (0.38) ALDH1A1HTR4
SCHEMBL5215519 0.80 HTR4 (0.33) HTR4GAA
SCHEMBL7446739 0.79 ITGB3 (0.40) ALDH1A1KDM4EHRH3MEN1KMT2A
SCHEMBL5219473 0.79 GNAO1 (0.38) ALDH1A1KDM4EMEN1KMT2AALOX15
SCHEMBL5218969 0.79 HTR4 (0.35) ALDH1A1KDM4EMEN1KMT2AHTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112270-B1 DIHYDROBENZODIOXINE CARBOXAMIDE AND KETONE DERIVATIVES AS 5-HT4 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2007-03-21 EP claimed
EP-1112270-B1 DIHYDROBENZODIOXINE CARBOXAMIDE AND KETONE DERIVATIVES AS 5-HT4 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed