SCHEMBL5218890

SCHEMBL5218890

Nc1nccc(Cc2ccc3ccccc3c2)c1N

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 3/20 0.52
MPO P05164 1/20 0.50
ALOX5 P09917 1/20 0.45
CYP2D6 P10635 1/20 0.43
NFKB1 P19838 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
PDE10A Q9Y233 1/20 0.42
BACE1 P56817 1/20 0.42
CTRC Q99895 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2A6 P11509 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27997631 0.84 ALDH1A1 (0.49) PDE10A
SCHEMBL7499087 0.80 LTA4H (0.43) ROCK1MPOBACE1
SCHEMBL31331676 0.80 ALOX5 (0.53) MPOALOX5CYP2D6NFKB1TAAR1
SCHEMBL5249618 0.78 MPO (0.46) MPOTAAR1
SCHEMBL5214698 0.76 DHFR (0.63) MPO
SCHEMBL9829477 0.75 DHFR (0.63)
SCHEMBL9536189 0.73 NOS2 (0.47) ROCK1
SCHEMBL3906522 0.73 MPO (0.43) MPOTAAR1
SCHEMBL9535888 0.73 ALDH1A1 (0.51) ROCK1MPOCYP2D6PDE10A
SCHEMBL5215491 0.73 F12 (0.53) CYP2D6TAAR1BACE1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831170-A1 SUBSTITUTED AMINOPYRIDINES AND USES THEREOF AstraZeneca AB (SE) 2007-09-12 EP disclosed
WO-2006065204-A1 SUBSTITUTED AMINOPYRIDINES AND USES THEREOF ASTRAZENECA AB (SE) 2006-06-22 WO disclosed