SCHEMBL5239176

SCHEMBL5239176

NC(=O)C[C@@H](c1ccccc1)N1CC2CN(C(=O)Cc3cccs3)CC2C1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.43
ALDH1A1 P00352 5/20 0.40
HSD17B10 Q99714 2/20 0.40
LMNA P02545 2/20 0.40
KDM4E B2RXH2 2/20 0.40
HPGD P15428 1/20 0.40
CASP1 P29466 1/20 0.40
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
PKM P14618 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
POLB P06746 2/20 0.39
TSHR P16473 1/20 0.39
NPC1 O15118 1/20 0.39
MAPT P10636 2/20 0.38
GFER P55789 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
GAA P10253 1/20 0.37
CASP6 P55212 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5240008 0.83 ALDH1A1 (0.48) HTTALDH1A1HSD17B10LMNAKDM4E
SCHEMBL5237872 0.81 CCL5 (0.40) ALDH1A1LMNAHPGDMEN1KMT2A
SCHEMBL4692754 0.77 HTT (0.46) HTTALDH1A1HSD17B10LMNAKDM4E
SCHEMBL5232470 0.73 CCR5 (0.54)
SCHEMBL5234052 0.72 PKM (0.46) HTTALDH1A1HSD17B10KDM4EHPGD
SCHEMBL5229817 0.72 CCR5 (0.42) ALDH1A1TDP1
SCHEMBL5235073 0.72 CHRNB2 (0.53) ALDH1A1SMN1; SMN2GAA
SCHEMBL5229656 0.72 CCR5 (0.40)
SCHEMBL5234982 0.71 CCR5 (0.42) HPGD
SCHEMBL5235854 0.70 PARP1 (0.37) HPGDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed