SCHEMBL5239767

SCHEMBL5239767

CNC1(CC=O)CN(c2ccccc2OCC(F)(F)F)CCN1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 9/20 0.40
ADRA1B P35368 9/20 0.40
ADRA1D P25100 8/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
DRD2 P14416 1/20 0.37
UGCG Q16739 1/20 0.36
SOAT1 P35610 1/20 0.35
GAA P10253 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5234068 0.86 DRD2 (0.45) CYP3A4CYP2C9CYP2C19DRD2
SCHEMBL5237575 0.85 RBP4 (0.43)
SCHEMBL5239721 0.84 TSHR (0.41) ADRA1AADRA1BADRA1DDRD2
SCHEMBL5239761 0.82 ADRA1A (0.41) ADRA1AADRA1BADRA1DCYP3A4CYP2C9
SCHEMBL5235916 0.81 AR (0.40) CYP2C9CYP2C19L3MBTL1
SCHEMBL5237871 0.81 DRD2 (0.40) DRD2GAA
SCHEMBL5238575 0.79 CXCR3 (0.38) ADRA1ADRD2
SCHEMBL5238192 0.78 CYP2C19 (0.37) CYP3A4CYP2C9CYP2C19
SCHEMBL5238831 0.77 ALDH1A1 (0.43) GAAL3MBTL1
SCHEMBL5235194 0.75 PKM (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1701946-B1 DERIVATIVES OF 1-PIPERAZINE- AND 1-HOMOPIPERAZINE-CARBOXYLATES, PREPARATION METHOD THEREOF AND USE OF SAME AS INHIBITORS OF THE FAAH ENZYME SANOFI AVENTIS (FR) 2007-12-19 EP claimed