SCHEMBL527664

SCHEMBL527664

O=C1CCc2ccc(Cl)nc21

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PBRM1 Q86U86 1/20 0.34
TDP2 O95551 1/20 0.34
NSD2 O96028 1/20 0.34
HTR1A P08908 2/20 0.33
HTR2A P28223 2/20 0.33
IDO1 P14902 1/20 0.32
DRD2 P14416 1/20 0.32
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29864428 1.00 PBRM1 (0.34) PBRM1TDP2NSD2HTR1AHTR2A
SCHEMBL30002194 0.88 MAOA (0.38) TDP2NSD2HTR1AHTR2AHSD17B10
SCHEMBL6635128 0.88 MAOA (0.38) TDP2NSD2HTR1AHTR2AHSD17B10
SCHEMBL12446468 0.84 HTR2A (0.33) TDP2NSD2HTR1AHTR2A
SCHEMBL10187270 0.79 CASP1 (0.38) PBRM1DRD2CASP1CASP7HSD17B10
SCHEMBL23376841 0.75 PBRM1 (0.38) PBRM1CASP1CASP7HSD17B10
SCHEMBL24858516 0.75 PBRM1 (0.34) PBRM1HTR1AHTR2ADRD2CASP1
SCHEMBL22852089 0.75 PBRM1 (0.34) PBRM1CASP1CASP7HSD17B10
SCHEMBL24490882 0.75 PBRM1 (0.34) PBRM1CASP1CASP7HSD17B10
SCHEMBL527206 0.75 S100A4 (0.42) PBRM1NSD2HTR1AHTR2ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 79 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260028363-A1 CHIRAL SYNTHESIS OF A TERTIARY ALCOHOL RECURIUM IP HOLDINGS LLC (US) 2026-01-29 US disclosed
US-20250361241-A1 HPK1 INHIBITOR AND MEDICAL USE THEREOF BETTA PHARMACEUTICALS CO., LTD. (CN) 2025-11-27 US disclosed
EP-4619406-A1 TRICYCLIC COMPOUNDS Schrödinger, Inc. (US) 2025-09-24 EP disclosed
US-12410204-B2 Chiral synthesis of a tertiary alcohol RECURIUM IP HOLDINGS, LLC (US) 2025-09-09 US disclosed
EP-4538274-A1 HPK1 INHIBITOR AND MEDICAL USE THEREOF Betta Pharmaceuticals Co., Ltd (CN) 2025-04-16 EP disclosed
US-20240228459-A1 WEE1 INHIBITORS AND USES THEREOF BOUNDLESS BIO, INC. 2024-07-11 US disclosed
US-20240228459-A1 WEE1 INHIBITORS AND USES THEREOF BOUNDLESS BIO, INC. 2024-07-11 US disclosed
US-20240228459-A1 WEE1 INHIBITORS AND USES THEREOF BOUNDLESS BIO, INC. 2024-07-11 US disclosed
WO-2024107393-A1 TRICYCLIC COMPOUNDS SCHRÖDINGER, INC. (US) 2024-05-23 WO disclosed
WO-2023237085-A1 HPK1 INHIBITOR AND MEDICAL USE THEREOF 贝达药业股份有限公司 2023-12-14 WO disclosed
WO-2012038521-A1 NOVEL MICROBIOCIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-03-29 WO disclosed
EP-2432555-A1 N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-d]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS Incyte Corporation (US) 2012-03-28 EP disclosed
WO-2012013754-A1 NOVEL MICROBIOCIDAL DIOXIME ETHER DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2012-02-02 WO disclosed
WO-2012013754-A1 NOVEL MICROBIOCIDAL DIOXIME ETHER DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2012-02-02 WO disclosed
WO-2012001107-A1 PIPERIDINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-05 WO disclosed
WO-2012001040-A1 NOVEL MICROBIOCIDAL DIOXIME ETHER DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-05 WO disclosed
US-20110130384-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-06-02 US disclosed
EP-2298731-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-03-23 EP disclosed
WO-2010135650-A1 N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-d]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS INCYTE CORPORATION (US) 2010-11-25 WO disclosed
US-20100298334-A1 N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-d]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS INCYTE CORPORATION 2010-11-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100298334-A1 N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-d]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS JAK1, JAK3, JAK2 PBRM1 263/4885TDP2 1495/4885NSD2 412/4885
US-12410204-B2 Chiral synthesis of a tertiary alcohol ADH1A, ADH1C, ADH5 PBRM1 354/4885TDP2 3952/4885NSD2 4763/4885
US-20250361241-A1 HPK1 INHIBITOR AND MEDICAL USE THEREOF STK11, STK35, STK10 PBRM1 897/4885TDP2 1776/4885NSD2 3004/4885
US-20110130384-A1 AMIDE COMPOUND GPR52, CNR2, ARRB1 PBRM1 2809/4885TDP2 3911/4885NSD2 1711/4885
US-20240228459-A1 WEE1 INHIBITORS AND USES THEREOF WEE1, WEE2, DCLRE1B PBRM1 1935/4885TDP2 386/4885NSD2 1908/4885
US-20260028363-A1 CHIRAL SYNTHESIS OF A TERTIARY ALCOHOL ADH1A, ADH1C, ADH5 PBRM1 236/4885TDP2 3449/4885NSD2 3612/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.