SCHEMBL5299686

SCHEMBL5299686

Nc1nsc(S(=O)(=O)Cc2ccccc2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA2B P29275 1/20 0.46
ADORA1 P30542 1/20 0.46
CYP2D6 P10635 1/20 0.45
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA5A P35218 1/20 0.43
CA9 Q16790 1/20 0.43
LOX P28300 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.43
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
HSD17B10 Q99714 2/20 0.41
KDM4E B2RXH2 1/20 0.41
PRSS1 P07477 2/20 0.39
PRSS2 P07478 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7513501 0.81 ADORA3 (0.46) ADORA3ADORA2AADORA2BADORA1CYP2D6
SCHEMBL5293941 0.77 TXNRD1 (0.43) CYP2D6CA1CA2CA5ACA9
SCHEMBL5303795 0.77 LOXL2 (0.48) ADORA3ADORA2AADORA2BADORA1LOXL2
SCHEMBL5363871 0.76 PLAU (0.41) ADORA3ADORA2AADORA2BADORA1CA1
SCHEMBL11328859 0.74 CYP2D6 (0.48) ADORA3ADORA2AADORA2BADORA1CYP2D6
SCHEMBL5306349 0.74 ALDH1A1 (0.43) CYP2D6ALDH1A1HSD17B10
SCHEMBL5368484 0.72 SMN1; SMN2 (0.43) CA1CA2CA5ACA9ALDH1A1
SCHEMBL9870797 0.72 KMT2A (0.51) CYP2D6CA1CA2CA5ACA9
SCHEMBL5298572 0.69 LOXL2 (0.36) LOXL2ALDH1A1HPGDLMNAKDM4E
SCHEMBL5288067 0.69 LOX (0.34) LOX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007012724-A1 1,2,4-THIADIAZOLE DERIVATIVES ANTIFUNGAL COMPOUNDS, COMPOSITIONS CONTAINING SAID COMPOUNDS AND THE USE THEREOF CYTOMICS SYSTEMS (FR) 2007-02-01 WO claimed
WO-2007012724-A1 1,2,4-THIADIAZOLE DERIVATIVES ANTIFUNGAL COMPOUNDS, COMPOSITIONS CONTAINING SAID COMPOUNDS AND THE USE THEREOF CYTOMICS SYSTEMS (FR) 2007-02-01 WO disclosed