SCHEMBL5322868

SCHEMBL5322868

COc1ccc(CNCC(O)Cn2c(=O)cc(-c3ccc(C)cc3)n(-c3ccc(SC)cc3)c2=O)c(OC)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
MAPT P10636 4/20 0.39
NPSR1 Q6W5P4 3/20 0.39
KMT2A Q03164 3/20 0.39
KDM4E B2RXH2 3/20 0.39
PDCD1 Q15116 2/20 0.36
CD274 Q9NZQ7 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
DNM1 Q05193 2/20 0.36
APLNR P35414 1/20 0.36
MITF O75030 1/20 0.36
LMNA P02545 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
MEN1 O00255 2/20 0.35
NR2F2 P24468 1/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTR2A P28223 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14622465 0.89 DNM1 (0.44) ALDH1A1MAPTKMT2AKDM4EDNM1
SCHEMBL5329856 0.82 DNM1 (0.45) ALDH1A1KMT2AKDM4ESMN1; SMN2DNM1
SCHEMBL5328787 0.79 DNM1 (0.44) ALDH1A1MAPTKMT2AKDM4ESMN1; SMN2
SCHEMBL5321578 0.78 PTGS2 (0.37) MAPTSMN1; SMN2APLNRLMNACYP2C9
SCHEMBL5323252 0.77 PTGS2 (0.35) MAPTSMN1; SMN2APLNRLMNACYP2C9
SCHEMBL5327487 0.75 DNM1 (0.34) MAPTSMN1; SMN2DNM1LMNACYP2C9
SCHEMBL14622407 0.75 PTGS2 (0.38) ALDH1A1MAPTNPSR1SMN1; SMN2LMNA
SCHEMBL5323331 0.74 RGS4 (0.48) ALDH1A1MAPTKDM4ESMN1; SMN2MITF
SCHEMBL5325599 0.73 KDM4E (0.38) ALDH1A1MAPTKMT2AKDM4ESMN1; SMN2
SCHEMBL5325697 0.73 RAD51 (0.40) SMN1; SMN2APLNRLMNACYP2C9HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO claimed
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed