SCHEMBL5325599

SCHEMBL5325599

CSc1ccc(-n2c(-c3ccc(C)cc3)cc(=O)n(CC(O)CN3CCN(C)CC3)c2=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
MAPT P10636 3/20 0.38
HTT P42858 2/20 0.38
RAD52 P43351 1/20 0.38
PRMT5 O14744 3/20 0.34
WDR77 Q9BQA1 3/20 0.34
ALDH1A1 P00352 3/20 0.34
HPGD P15428 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
MAPK1 P28482 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
ABCB1 P08183 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5321659 0.90 ALOX15 (0.43) KDM4EMEN1KMT2AMAPTHTT
SCHEMBL14622410 0.89 MAPT (0.43) KDM4EMEN1KMT2AMAPTHTT
SCHEMBL5323186 0.86 MAPT (0.51) KDM4EMEN1KMT2AMAPTHTT
SCHEMBL5321578 0.85 PTGS2 (0.37) MAPTHTTSMN1; SMN2LMNAPTGS2
SCHEMBL5325651 0.85 LMNA (0.47) KDM4EMEN1KMT2AMAPTHTT
SCHEMBL5323252 0.84 PTGS2 (0.35) MAPTHTTSMN1; SMN2LMNAMAPK1
SCHEMBL5327487 0.83 DNM1 (0.34) MAPTHTTSMN1; SMN2LMNAPTGS2
SCHEMBL14622908 0.82 DRD2 (0.38)
SCHEMBL5325610 0.81 MEN1 (0.39) KDM4EMEN1KMT2AMAPTHTT
SCHEMBL14622407 0.80 PTGS2 (0.38) MAPTHTTALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed