SCHEMBL5328645

SCHEMBL5328645

COc1ccc(CS(=O)(=O)c2nc(CSc3ccc(C)cc3)ns2)cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 6/20 0.37
MAPK1 P28482 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
PPARD Q03181 3/20 0.35
PPARA Q07869 2/20 0.35
LMNA P02545 2/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
MAOB P27338 1/20 0.35
MEN1 O00255 1/20 0.35
GFER P55789 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5293270 0.83 ALDH1A1 (0.37) SMN1; SMN2NPC1RAB9AALDH1A1MAPK1
SCHEMBL5328644 0.77 SMN1; SMN2 (0.37) SMN1; SMN2NPC1RAB9AALDH1A1MAPK1
SCHEMBL5291890 0.71 PPARD (0.41) SMN1; SMN2RAB9APPARDPPARALMNA
SCHEMBL5298909 0.68 POLB (0.45) ALDH1A1L3MBTL1HTTMAPTKMT2A
SCHEMBL7535556 0.65 TUBB1 (0.43) SMN1; SMN2NPC1RAB9AALDH1A1MAPK1
SCHEMBL29665700 0.65 TUBB1 (0.43) SMN1; SMN2NPC1RAB9AALDH1A1MAPK1
SCHEMBL8793443 0.63 CA2 (0.52) SMN1; SMN2ALDH1A1PPARDPPARALMNA
SCHEMBL30745833 0.63 LMNA (0.48) SMN1; SMN2RAB9AALDH1A1MAPK1LMNA
SCHEMBL5298171 0.62 TXNRD1 (0.45) SMN1; SMN2ALDH1A1MAPK1L3MBTL1LMNA
SCHEMBL24458142 0.62 TUBB1 (0.39) RAB9AALDH1A1MAPK1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007012724-A1 1,2,4-THIADIAZOLE DERIVATIVES ANTIFUNGAL COMPOUNDS, COMPOSITIONS CONTAINING SAID COMPOUNDS AND THE USE THEREOF CYTOMICS SYSTEMS (FR) 2007-02-01 WO disclosed